SCHEMBL28558865

SCHEMBL28558865

Fc1cc(-c2n[nH]c3ncc(Br)cc23)c(Cl)cn1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 5/20 0.34
DYRK1B Q9Y463 5/20 0.34
AURKA O14965 3/20 0.34
JAK2 O60674 3/20 0.34
MAP4K4 O95819 3/20 0.34
FGFR1 P11362 3/20 0.34
FLT1 P17948 3/20 0.34
KDR P35968 3/20 0.34
CLK2 P49760 3/20 0.34
CDK5 Q00535 3/20 0.34
MAP4K2 Q12851 3/20 0.34
AURKB Q96GD4 3/20 0.34
CLK4 Q9HAZ1 3/20 0.34
IGF1R P08069 2/20 0.34
JAK3 P52333 2/20 0.34
LIMK1 P53667 2/20 0.34
NTRK2 Q16620 2/20 0.34
DAPK3 O43293 2/20 0.34
PAK4 O96013 2/20 0.34
ABL1 P00519 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28607892 0.77 DYRK1A (0.52) DYRK1ADYRK1BAURKAJAK2MAP4K4
SCHEMBL28556801 0.76 IDO1 (0.44) DYRK1ADYRK1BAURKAJAK2MAP4K4
SCHEMBL28549353 0.72 KIT (0.45) DYRK1ADYRK1BAURKAJAK2MAP4K4
SCHEMBL16537147 0.71 DYRK1B (0.44) DYRK1ADYRK1BAURKAJAK2MAP4K4
SCHEMBL28553148 0.69 DYRK1B (0.56) DYRK1ADYRK1BAURKAJAK2MAP4K4
SCHEMBL5061384 0.69 DYRK1A (0.57) DYRK1ADYRK1BAURKAJAK2MAP4K4
SCHEMBL28559332 0.68 DYRK1A (0.44) DYRK1ADYRK1BAURKAJAK2MAP4K4
SCHEMBL22820704 0.68 KMT2A (0.43) DYRK1AMAP4K4MINK1MET
SCHEMBL29930538 0.68 DYRK1B (0.60) DYRK1ADYRK1BAURKAJAK2MAP4K4
SCHEMBL29930770 0.67 DYRK1B (0.58) DYRK1ADYRK1BAURKAJAK2MAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112724134-B Azaindazole bipyridine derivative myeloid cell proliferation inhibitor, preparation method and application thereof in pharmacy 复旦大学 2022-04-01 CN disclosed
CN-112724134-A Azaindazole bipyridine derivative myeloid cell proliferation inhibitor, preparation method and application thereof in pharmacy 复旦大学 2021-04-30 CN disclosed