SCHEMBL28560474

SCHEMBL28560474

CC(C)(C)OC(=O)N1CCC(Oc2c(OC3CCOC3)ccc(Br)c2C#N)C(F)(F)C1

nearest known ligand 0.37

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 4/20 0.37
TBK1 Q9UHD2 6/20 0.36
PDE4B Q07343 5/20 0.35
PDE4D Q08499 5/20 0.35
PDE4A P27815 3/20 0.34
PDE4C Q08493 3/20 0.34
ALK Q9UM73 2/20 0.33
SLC6A9 P48067 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30988767 1.00 GPR119 (0.37) GPR119TBK1PDE4BPDE4DPDE4A
SCHEMBL21886828 1.00 GPR119 (0.37) GPR119TBK1PDE4BPDE4DPDE4A
SCHEMBL25987132 0.88 PDE4B (0.40) GPR119PDE4BPDE4DPDE4APDE4C
SCHEMBL25987087 0.85 GPR119 (0.36) GPR119TBK1PDE4BPDE4DPDE4A
SCHEMBL30988791 0.85 GPR119 (0.37) GPR119PDE4BPDE4DPDE4APDE4C
SCHEMBL28555129 0.83 ERBB2 (0.39) TBK1PDE4BPDE4DPDE4APDE4C
SCHEMBL21886826 0.83 GPR119 (0.40) GPR119ALK
SCHEMBL21886628 0.83 ERBB2 (0.39) TBK1PDE4BPDE4DPDE4APDE4C
SCHEMBL21886730 0.79 CHEK1 (0.38) PDE4BPDE4DPDE4APDE4C
SCHEMBL28559957 0.79 CHEK1 (0.38) PDE4BPDE4DPDE4APDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118255772-A Quinazoline derivatives as antitumor agents 苏州赞荣医药科技有限公司 2024-06-28 CN disclosed
CN-112654612-A Quinazoline derivatives as antitumor agents 苏州赞荣医药科技有限公司 2021-04-13 CN disclosed