SCHEMBL28555129

SCHEMBL28555129

CN1CCC(Oc2c(OC3CCOC3)ccc(Br)c2C#N)C(F)(F)C1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 3/20 0.39
EGFR P00533 1/20 0.39
IKBKE Q14164 3/20 0.34
TBK1 Q9UHD2 3/20 0.34
ALK Q9UM73 1/20 0.32
CHEK1 O14757 2/20 0.32
PDE4B Q07343 4/20 0.31
PDE4D Q08499 6/20 0.31
PDE4A P27815 3/20 0.31
PDE4C Q08493 3/20 0.31
MAPK8 P45983 1/20 0.31
MAPK9 P45984 1/20 0.31
EPHA2 P29317 1/20 0.31
KDR P35968 1/20 0.31
EPHB4 P54760 1/20 0.31
PDE9A O76083 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21886628 1.00 ERBB2 (0.39) ERBB2EGFRIKBKETBK1ALK
SCHEMBL28564240 0.89 EGFR (0.37) ERBB2EGFRIKBKETBK1ALK
SCHEMBL21886669 0.89 EGFR (0.37) ERBB2EGFRIKBKETBK1ALK
SCHEMBL25987137 0.85 ERBB2 (0.38) ERBB2EGFRTBK1CHEK1
SCHEMBL28569856 0.85 PDE4D (0.36) ERBB2EGFRCHEK1PDE4BPDE4D
SCHEMBL28569853 0.85 PDE4D (0.36) ERBB2EGFRCHEK1PDE4BPDE4D
SCHEMBL21886635 0.84 EGFR (0.35) ERBB2EGFRIKBKETBK1CHEK1
SCHEMBL21886828 0.83 GPR119 (0.37) TBK1ALKPDE4BPDE4DPDE4A
SCHEMBL30988767 0.83 GPR119 (0.37) TBK1ALKPDE4BPDE4DPDE4A
SCHEMBL28560474 0.83 GPR119 (0.37) TBK1ALKPDE4BPDE4DPDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118255772-A Quinazoline derivatives as antitumor agents 苏州赞荣医药科技有限公司 2024-06-28 CN disclosed
CN-112654612-A Quinazoline derivatives as antitumor agents 苏州赞荣医药科技有限公司 2021-04-13 CN disclosed