SCHEMBL28564133

SCHEMBL28564133

Cc1ccc(N=C=O)c(F)c1F

nearest known ligand 0.50

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.50
TRPA1 O75762 1/20 0.50
HPGD P15428 2/20 0.39
ALDH1A1 P00352 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
GABRA1 P14867 1/20 0.31
GABRB2 P47870 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28566853 0.82 CYP3A4 (0.46) CYP3A4TRPA1HPGDALDH1A1TDP1
SCHEMBL27985693 0.82 CYP3A4 (0.61) CYP3A4TRPA1HPGDALDH1A1TDP1
SCHEMBL17650560 0.79 ALDH1A1 (0.37) CYP3A4HPGDALDH1A1TDP1GABRA1
SCHEMBL162877 0.78 CYP3A4 (0.40) CYP3A4TRPA1HPGDALDH1A1TDP1
SCHEMBL30438482 0.78 CYP3A4 (0.40) CYP3A4TRPA1HPGDALDH1A1TDP1
SCHEMBL28554406 0.75 TDP1 (0.44) CYP3A4TRPA1HPGDALDH1A1TDP1
SCHEMBL27699035 0.75 CYP3A4 (0.56) CYP3A4TRPA1HPGDALDH1A1TDP1
SCHEMBL29606267 0.74 CYP3A4 (0.61) CYP3A4TRPA1HPGDALDH1A1TDP1
SCHEMBL11608345 0.74 CYP3A4 (0.61) CYP3A4TRPA1HPGDALDH1A1TDP1
SCHEMBL1022418 0.73 CYP3A4 (0.63) CYP3A4TRPA1HPGDALDH1A1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113248506-A Substituted aminopurine compounds, compositions thereof, and methods of treatment therewith 西格诺药品有限公司 2021-08-13 CN disclosed
CN-107001372-B Substituted aminopurine compounds, compositions thereof, and methods of treatment therewith 西格诺药品有限公司 2021-04-27 CN disclosed