SCHEMBL28564602

SCHEMBL28564602

CC(C)(C)OC(Cc1ccc(Br)cc1)C(N)=O

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 4/20 0.45
MME P08473 2/20 0.43
PPARG P37231 2/20 0.43
PPARA Q07869 2/20 0.43
CTSS P25774 1/20 0.41
CTSK P43235 1/20 0.41
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
ACACB O00763 1/20 0.38
PPARD Q03181 1/20 0.38
MMP1 P03956 2/20 0.37
HDAC1 Q13547 2/20 0.36
HDAC6 Q9UBN7 2/20 0.36
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28571792 0.79 LMNA (0.44) EPHX1MMEPPARGPPARACTSS
SCHEMBL28598197 0.76 CTSS (0.45) EPHX1MMEPPARGCTSSCTSK
SCHEMBL2720266 0.73 EPHX1 (0.57) EPHX1MMEMEN1KMT2AACACB
SCHEMBL13643239 0.73 EPHX1 (0.57) EPHX1MMEMEN1KMT2AACACB
SCHEMBL8310103 0.73 CTSS (0.67) CTSSCTSK
SCHEMBL2617401 0.73 CTSS (0.67) CTSSCTSK
SCHEMBL7340685 0.72 CTSS (0.47) EPHX1MMECTSSCTSKACACB
SCHEMBL10562986 0.72 CTSS (0.47) EPHX1MMECTSSCTSKACACB
SCHEMBL4072985 0.72 MME (0.43) EPHX1MMEPPARGPPARACTSS
SCHEMBL7328879 0.72 CA1 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112661671-B Preparation method of Sacubitril intermediate 江苏阿尔法药业股份有限公司 2022-04-22 CN disclosed
CN-112661671-A Preparation method of Sacubitril intermediate 江苏阿尔法药业有限公司 2021-04-16 CN disclosed