SCHEMBL28565280

SCHEMBL28565280

O=CC1c2ccccc2C=CN1c1ccccn1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.34
BRD4 O60885 1/20 0.34
CCL2 P13500 1/20 0.34
TSHR P16473 2/20 0.33
NPSR1 Q6W5P4 1/20 0.33
LMNA P02545 2/20 0.33
MAPT P10636 2/20 0.33
CRBN Q96SW2 1/20 0.33
EP300 Q09472 1/20 0.33
KAT2B Q92831 1/20 0.33
ALDH1A1 P00352 4/20 0.32
KDM4E B2RXH2 3/20 0.32
GAA P10253 3/20 0.32
CYP1A2 P05177 2/20 0.32
MAPK1 P28482 2/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
HPGD P15428 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16245516 0.77 BRD4 (0.38) BRD4CCL2MAPTALDH1A1KDM4E
SCHEMBL28089129 0.72 BRD4 (0.49) SMN1; SMN2BRD4CCL2LMNAMAPT
SCHEMBL29290952 0.71 SMN1; SMN2 (0.41) SMN1; SMN2MAPTCRBNEP300KAT2B
SCHEMBL28147769 0.71 BRD4 (0.37) BRD4CCL2MAPTALDH1A1KDM4E
SCHEMBL29290947 0.71 SMN1; SMN2 (0.41) SMN1; SMN2MAPTCRBNEP300KAT2B
SCHEMBL28099962 0.71 CRBN (0.35) SMN1; SMN2MAPTCRBNEP300KAT2B
SCHEMBL28209858 0.71 SMN1; SMN2 (0.34) SMN1; SMN2TSHRNPSR1LMNACRBN
Hydrochloric Acid SCHEMBL27913881 0.70 BRD4 (0.47) SMN1; SMN2BRD4CCL2LMNAMAPT
SCHEMBL27682027 0.70 BRD4 (0.40) BRD4CCL2MAPTALDH1A1CYP1A2
SCHEMBL29290943 0.69 KDM4E (0.36) SMN1; SMN2TSHRLMNACRBNEP300

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109942542-B Preparation method of 3- (1, 3-diene-2-yl) isoquinoline-1 (2H) -ketone compound 南开大学 2021-05-07 CN disclosed