SCHEMBL2856684

SCHEMBL2856684

COc1ccc(CNC(=O)c2cnn(C)c2Cl)c(OC)c1

nearest known ligand 0.58

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 2/20 0.58
TAS1R1 Q7RTX1 2/20 0.58
ALDH1A1 P00352 2/20 0.56
TSHR P16473 1/20 0.56
NPSR1 Q6W5P4 1/20 0.56
GAA P10253 1/20 0.56
PKM P14618 1/20 0.56
HPGD P15428 1/20 0.56
HTT P42858 1/20 0.56
KLKB1 P03952 1/20 0.54
PDE4B Q07343 1/20 0.52
TP53 P04637 2/20 0.50
MAPT P10636 3/20 0.49
MAOB P27338 1/20 0.49
THRB P10828 1/20 0.48
KDM4C Q9H3R0 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24914439 0.80 TAS1R3 (0.66) TAS1R3TAS1R1ALDH1A1TSHRNPSR1
SCHEMBL29950449 0.79 BCDIN3D (0.51) TAS1R3TAS1R1ALDH1A1TSHRNPSR1
SCHEMBL27028480 0.79 BCDIN3D (0.51) TAS1R3TAS1R1ALDH1A1TSHRNPSR1
SCHEMBL23115900 0.79 TSHR (0.54) TAS1R3TAS1R1ALDH1A1TSHRNPSR1
SCHEMBL29766092 0.79 TSHR (0.54) TAS1R3TAS1R1ALDH1A1TSHRNPSR1
SCHEMBL703591 0.79 ALDH1A1 (0.56) TAS1R3TAS1R1ALDH1A1TSHRNPSR1
SCHEMBL23985899 0.79 TAS1R3 (0.71) TAS1R3TAS1R1ALDH1A1TSHRNPSR1
SCHEMBL30305533 0.79 TAS1R3 (0.71) TAS1R3TAS1R1ALDH1A1TSHRNPSR1
SCHEMBL2850378 0.79 EZH2 (0.46) ALDH1A1HPGDHTTTP53MAPT
SCHEMBL23115839 0.78 ALDH1A1 (0.64) TAS1R3TAS1R1ALDH1A1TSHRNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP disclosed