SCHEMBL28566867

SCHEMBL28566867

CCc1ccc(C#N)c(CC)c1Cl

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AR P10275 10/20 0.38
TRPV4 Q9HBA0 1/20 0.33
CTRC Q99895 1/20 0.33
KDM4E B2RXH2 3/20 0.33
ALDH1A1 P00352 2/20 0.33
LMNA P02545 2/20 0.33
KDM5A P29375 2/20 0.33
HPGD P15428 2/20 0.33
HSD17B10 Q99714 1/20 0.33
MEN1 O00255 1/20 0.33
GAA P10253 1/20 0.33
KMT2A Q03164 1/20 0.33
VCAM1 P19320 1/20 0.33
CYP2A6 P11509 1/20 0.32
NOS3 P29474 2/20 0.32
NOS1 P29475 2/20 0.32
NOS2 P35228 2/20 0.32
L3MBTL1 Q9Y468 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10878832 0.86 AR (0.45) ARTRPV4CYP2A6
SCHEMBL11514426 0.82 CYP2A6 (0.35) ARTRPV4KDM4EALDH1A1LMNA
SCHEMBL28574963 0.78 AR (0.36) ARTRPV4KDM4EALDH1A1LMNA
SCHEMBL28571188 0.77 PGR (0.33) ARKDM4EALDH1A1LMNAKDM5A
SCHEMBL12763627 0.77 AR (0.50) AR
SCHEMBL28571837 0.76 TRPV4 (0.44) ARTRPV4KDM4EGAAVCAM1
SCHEMBL28200532 0.76 AR (0.41) ARTRPV4CTRCKDM4EALDH1A1
SCHEMBL18552713 0.76 AR (0.44) ARVCAM1
SCHEMBL31352954 0.74 KDM4E (0.33) ARKDM4EALDH1A1LMNAKDM5A
SCHEMBL12763867 0.74 KDM5A (0.36) ARKDM4EALDH1A1LMNAKDM5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112778215-A 2-methoxyphenoxy pyrimidine antitumor compound and preparation method and application thereof 中国医科大学 2021-05-11 CN disclosed