SCHEMBL28566904

SCHEMBL28566904

O=C(O)c1cc2cccnc2nc1Cc1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.45
KDM4E B2RXH2 3/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
ALDH1A1 P00352 4/20 0.43
CYP2C9 P11712 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
KDM4A O75164 1/20 0.42
KDM5A P29375 1/20 0.42
KDM4C Q9H3R0 1/20 0.42
KDM5B Q9UGL1 1/20 0.42
HNF4A P41235 1/20 0.41
MCL1 Q07820 1/20 0.41
PTPN1 P18031 3/20 0.40
ALOX12 P18054 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
EGLN1 Q9GZT9 1/20 0.40
ACMSD Q8TDX5 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28550680 0.82 KDM4E (0.47) LMNAKDM4EMEN1KMT2AALDH1A1
SCHEMBL258223 0.77 ALDH1A1 (0.55) LMNAKDM4EALDH1A1CYP2C9SMN1; SMN2
SCHEMBL7278161 0.75 KDM4E (0.55) LMNAKDM4EMEN1KMT2AALDH1A1
SCHEMBL352470 0.75 KDM4E (0.53) LMNAKDM4EMEN1KMT2AALDH1A1
SCHEMBL253870 0.75 CYP11B1 (0.52) NPC1CYP3A4
SCHEMBL17942663 0.75 DHODH (0.51) LMNAKDM4EMEN1KMT2AALDH1A1
SCHEMBL125290 0.74 LMNA (0.51) LMNAKDM4EMEN1KMT2AALDH1A1
SCHEMBL27836545 0.74 LMNA (0.56) LMNAKDM4EMEN1KMT2AALDH1A1
SCHEMBL252393 0.74 LMNA (0.47) LMNAKDM4EMEN1KMT2AALDH1A1
SCHEMBL253705 0.73 AURKA (0.47) CYP2C9CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112752762-A Substituted pyridoindoles for the treatment and prevention of bacterial infections 豪夫迈·罗氏有限公司 2021-05-04 CN disclosed