SCHEMBL28568917

SCHEMBL28568917

Brc1nnnnc1-c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 5/20 0.48
HTT P42858 2/20 0.48
ALOX15 P16050 1/20 0.42
MAPK1 P28482 4/20 0.42
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
ALDH1A1 P00352 4/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
XDH P47989 1/20 0.40
MAPT P10636 1/20 0.40
ADORA2A P29274 1/20 0.40
ADORA1 P30542 1/20 0.40
CLK4 Q9HAZ1 2/20 0.39
CSNK1A1 P48729 1/20 0.39
PDE5A O76074 2/20 0.39
PDE1A P54750 2/20 0.39
PDE1B Q01064 2/20 0.39
PDE3B Q13370 2/20 0.39
PDE1C Q14123 2/20 0.39
PDE3A Q14432 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7197255 0.84 LMNA (0.56) LMNAHTTALOX15MAPK1NPC1
SCHEMBL29516583 0.75 LMNA (0.48) LMNAHTTALOX15MAPK1NPC1
SCHEMBL24501024 0.74 LMNA (0.50) LMNAHTTALOX15MAPK1ALDH1A1
SCHEMBL28214061 0.73 LMNA (0.42) LMNAHTTALOX15MAPK1NPC1
SCHEMBL500715 0.72 LMNA (0.56) LMNAHTTALOX15MAPK1NPC1
SCHEMBL27990057 0.72 ADORA2A (0.68) XDHADORA2AADORA1CLK4CSNK1A1
SCHEMBL17287226 0.72 ALDH1A1 (0.54) LMNAHTTMAPK1NPC1RAB9A
Formamide SCHEMBL28090638 0.71 ADORA2A (0.47) LMNAHTTALOX15MAPK1NPC1
SCHEMBL22360955 0.70 LMNA (0.54) LMNAHTTALOX15MAPK1NPC1
SCHEMBL31637095 0.70 LMNA (0.46) LMNAHTTALOX15MAPK1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112812074-B Tetrazine compound and preparation method and application thereof 四川大学华西医院 2022-06-14 CN disclosed
CN-112812074-A Tetrazine compound and preparation method and application thereof 四川大学华西医院 2021-05-18 CN disclosed