SCHEMBL28569296

SCHEMBL28569296

Nc1cc(C(=O)O)cc(Br)c1N1CCCC(O)C1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.42
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.42
KDM4E B2RXH2 4/20 0.41
GAA P10253 3/20 0.41
HSD17B10 Q99714 2/20 0.41
POLB P06746 2/20 0.41
TDP1 Q9NUW8 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
NR4A1 P22736 1/20 0.38
SMARCA2 P51531 1/20 0.37
SMARCA4 P51532 1/20 0.37
PBRM1 Q86U86 1/20 0.37
SMPD3 Q9NY59 2/20 0.36
IKBKB O14920 2/20 0.36
TTR P02766 1/20 0.35
HDAC6 Q9UBN7 1/20 0.34
CCNE2 O96020 1/20 0.33
CCNE1 P24864 1/20 0.33
CDK2 P24941 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21808141 1.00 ALDH1A1 (0.42) ALDH1A1KMT2AMEN1KDM4EGAA
SCHEMBL21820524 0.85 NPC1 (0.45) ALDH1A1KDM4EGAAHSD17B10SMARCA2
SCHEMBL21820522 0.85 NPC1 (0.45) ALDH1A1KDM4EGAAHSD17B10SMARCA2
SCHEMBL21808171 0.82 KDM4E (0.55) ALDH1A1KMT2AMEN1KDM4EGAA
SCHEMBL28573261 0.81 ALDH1A1 (0.64) ALDH1A1KMT2AMEN1KDM4EGAA
SCHEMBL28573263 0.81 ALDH1A1 (0.64) ALDH1A1KMT2AMEN1KDM4EGAA
SCHEMBL28562860 0.77 KMT2A (0.37) ALDH1A1KMT2AMEN1KDM4EGAA
SCHEMBL28569424 0.72 GFER (0.43) ALDH1A1KMT2AMEN1KDM4EGAA
SCHEMBL21808119 0.72 GFER (0.43) ALDH1A1KMT2AMEN1KDM4EGAA
SCHEMBL1663436 0.69 USP2 (0.55) ALDH1A1KDM4EGAAHSD17B10L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115448908-A Compounds for the treatment of specific leukemias 拓臻股份有限公司 2022-12-09 CN disclosed
CN-115215838-A Compounds for the treatment of specific leukemias 拓臻股份有限公司 2022-10-21 CN disclosed
CN-112770745-B Compounds for the treatment of specific leukemias 拓臻股份有限公司 2022-09-02 CN disclosed
CN-112770745-A Compounds for the treatment of specific leukemias 拓臻股份有限公司 2021-05-07 CN disclosed