SCHEMBL28569504

SCHEMBL28569504

Nc1cc(Cc2ccc(Cl)cc2)[nH]n1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 1/20 0.56
MKNK2 Q9HBH9 1/20 0.56
LTA4H P09960 1/20 0.47
MPO P05164 1/20 0.47
HSP90AB1 P08238 1/20 0.45
DAO P14920 2/20 0.44
KDR P35968 1/20 0.43
NPC1 O15118 1/20 0.41
MAPT P10636 1/20 0.41
RAB9A P51151 1/20 0.41
GFER P55789 1/20 0.41
ALDH1A1 P00352 2/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
HPGD P15428 1/20 0.40
TSHR P16473 1/20 0.40
HCAR2 Q8TDS4 1/20 0.40
NR1H2 P55055 1/20 0.40
LMNA P02545 1/20 0.40
ALPL P05186 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17967278 0.84 MKNK1 (0.54) MKNK1MKNK2LTA4HMPODAO
SCHEMBL3499891 0.81 HPGD (0.59) MPOKDRGFERALDH1A1MEN1
Hydrochloric Acid SCHEMBL17397945 0.80 HPGD (0.57) MPOKDRGFERALDH1A1MEN1
SCHEMBL4853841 0.78 DYRK1A (0.59) LTA4HMPOKDRNPC1MAPT
SCHEMBL3259505 0.72 SCN9A (0.41) DAONPC1MAPTRAB9AALDH1A1
SCHEMBL5630086 0.72 MKNK1 (1.00) MKNK1MKNK2LTA4HNPC1MAPT
SCHEMBL13737504 0.71 HSP90AB1 (0.53) MKNK1MKNK2MPOHSP90AB1DAO
SCHEMBL3937754 0.68 MAPT (0.49) MPODAONPC1MAPTRAB9A
SCHEMBL10284906 0.68 HSP90AB1 (0.45) HSP90AB1DAONPC1MAPTRAB9A
SCHEMBL459184 0.68 LMNA (0.50) MKNK1MKNK2MPOHSP90AB1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112876482-B Polysubstituted heterocyclic derivative, preparation method and medical application thereof 中国药科大学 2023-07-28 CN disclosed
CN-112876482-A Polysubstituted heterocyclic derivative, preparation method and medical application thereof 中国药科大学 2021-06-01 CN disclosed