SCHEMBL459184

SCHEMBL459184

Nc1[nH]nc(Cc2ccc(Cl)cc2)c1N

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.50
ALDH1A1 P00352 2/20 0.41
HSP90AB1 P08238 1/20 0.41
MPO P05164 1/20 0.40
GAA P10253 2/20 0.39
MEN1 O00255 1/20 0.39
MAPT P10636 1/20 0.39
MAPK1 P28482 1/20 0.39
KMT2A Q03164 1/20 0.39
PARP1 P09874 1/20 0.37
NR1H2 P55055 1/20 0.36
MKNK1 Q9BUB5 1/20 0.36
MKNK2 Q9HBH9 1/20 0.36
ALPL P05186 1/20 0.36
GFER P55789 1/20 0.36
TAAR1 Q96RJ0 1/20 0.35
NOTUM Q6P988 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6241862 0.82 RECQL (0.41) LMNAALDH1A1GAAMEN1MAPT
SCHEMBL6240087 0.81 PARP1 (0.50) LMNAALDH1A1MPOPARP1NR1H2
SCHEMBL4625227 0.78 ALDH1A1 (0.53) LMNAALDH1A1MPOGAAMEN1
SCHEMBL20767297 0.74 NR1H2 (0.50) LMNAALDH1A1GAAMEN1MAPT
SCHEMBL13516409 0.72 P2RX7 (0.45) LMNAALDH1A1HSP90AB1MPOGAA
SCHEMBL4697722 0.68 LMNA (0.68) LMNAALDH1A1MEN1KMT2APARP1
SCHEMBL8012674 0.68 ALDH1A1 (0.41) LMNAALDH1A1HSP90AB1MPOGAA
SCHEMBL28569504 0.68 MKNK1 (0.56) LMNAALDH1A1HSP90AB1MPOMEN1
SCHEMBL13737504 0.68 HSP90AB1 (0.53) LMNAALDH1A1HSP90AB1MPOGAA
SCHEMBL8108506 0.67 ROCK2 (0.44) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 167 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1453476-A1 NOVEL OXIDATION DYES COMPRISING 2,4-DICHLORO-3-AMINOPHENOL Henkel Kommanditgesellschaft auf Aktien (DE) 2004-09-08 EP claimed
EP-1453477-A1 NOVEL DEVELOPER-COUPLER COMBINATION CONTAINING 2,4-DICHLORO-3-AMINOPHENOL Henkel Kommanditgesellschaft auf Aktien (DE) 2004-09-08 EP claimed
EP-1443889-A1 OXIDATION COLOURING AGENT BASED ON BICYCLIC DEVELOPER COMPONENTS Henkel Kommanditgesellschaft auf Aktien (DE) 2004-08-11 EP claimed
JP-3538424-B2 2004-06-14 JP claimed
EP-1367983-A1 MICROCAPSULES WITH AQUEOUS CORE CONTAINING OXIDATION-REDUCTION ENZYMES AND THEIR USE IN OXIDATION DYEING COMPOSITIONS L'OREAL (FR) 2003-12-10 EP claimed
WO-2003053384-A1 NOVEL DEVELOPER-COUPLER COMBINATION CONTAINING 2,4-DICHLORO-3-AMINOPHENOL HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 2003-07-03 WO claimed
WO-2003053385-A1 NOVEL OXIDATION DYES COMPRISING 2,4-DICHLORO-3-AMINOPHENOL HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 2003-07-03 WO claimed
WO-2003041672-A1 OXIDATION COLOURING AGENT BASED ON BICYCLIC DEVELOPER COMPONENTS HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 2003-05-22 WO claimed
WO-2002069922-A1 MICROCAPSULES WITH AQUEOUS CORE CONTAINING OXIDATION-REDUCTION ENZYMES AND THEIR USE IN OXIDATION DYEING COMPOSITIONS L'OREAL (FR) 2002-09-12 WO claimed
EP-1235550-A2 NEW COLOURING COMBINATION Henkel Kommanditgesellschaft auf Aktien (DE) 2002-09-04 EP claimed
WO-2001041717-A2 NEW COLOURING COMBINATION HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 2001-06-14 WO claimed
EP-0618903-A1 OXIDATION HAIR DYE CONTAINING 4,5-DIAMINOPYRAZOLE DERIVATIVES AND NOVEL 4,5-DIAMINOPYRAZOLE DERIVATIVES AND PROCESS FOR THEIR PRODUCTION Wella Aktiengesellschaft (DE) 1994-10-12 EP claimed
WO-1994008970-A1 OXIDATION HAIR DYE CONTAINING 4,5-DIAMINOPYRAZOLE DERIVATIVES AND NOVEL 4,5-DIAMINOPYRAZOLE DERIVATIVES AND PROCESS FOR THEIR PRODUCTION WELLA AKTIENGESELLSCHAFT (DE) 1994-04-28 WO claimed
EP-4642425-A1 COMPOSITION COMPRISING AT LEAST N,N-DICARBOXYMETHYLGLUTAMIC ACID, AT LEAST ONE COLOURING AGENT AND AT LEAST ONE FATTY AMINE L'OREAL (FR) 2025-11-05 EP disclosed
EP-4452214-A1 COMPOSITION FOR KERATIN FIBERS L'OREAL (FR) 2024-10-30 EP disclosed
WO-2024141615-A1 COMPOSITION COMPRISING AT LEAST N,N-DICARBOXYMETHYLGLUTAMIC ACID, AT LEAST ONE COLOURING AGENT AND AT LEAST ONE FATTY AMINE L'OREAL (FR) 2024-07-04 WO disclosed
WO-2000078273-A2 PROCESS FOR PRODUCING A HAIRDYE COMPOSITION LION CORPORATION (JP) 2000-12-28 WO disclosed
WO-2000057848-A1 OXIDATION DYEING METHOD USING N-ACETYLCYSTEINE AS A REDUCING AGENT AND LACCASE AS AN OXIDATING AGENT L'OREAL (FR) 2000-10-05 WO disclosed
EP-0618903-A1 OXIDATION HAIR DYE CONTAINING 4,5-DIAMINOPYRAZOLE DERIVATIVES AND NOVEL 4,5-DIAMINOPYRAZOLE DERIVATIVES AND PROCESS FOR THEIR PRODUCTION Wella Aktiengesellschaft (DE) 1994-10-12 EP disclosed
WO-1994008970-A1 OXIDATION HAIR DYE CONTAINING 4,5-DIAMINOPYRAZOLE DERIVATIVES AND NOVEL 4,5-DIAMINOPYRAZOLE DERIVATIVES AND PROCESS FOR THEIR PRODUCTION WELLA AKTIENGESELLSCHAFT (DE) 1994-04-28 WO disclosed