SCHEMBL28573282

SCHEMBL28573282

CCOC(=O)c1ccc(Nc2nnc(-c3ccccc3)s2)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 1/20 0.64
RARA P10276 1/20 0.57
RARB P10826 1/20 0.57
RARG P13631 1/20 0.57
NPC1 O15118 4/20 0.57
MEN1 O00255 3/20 0.57
KMT2A Q03164 3/20 0.57
GBA1 P04062 1/20 0.57
DHODH Q02127 5/20 0.56
MAPT P10636 5/20 0.56
RXFP1 Q9HBX9 2/20 0.55
LMNA P02545 2/20 0.55
POLB P06746 2/20 0.55
RAB9A P51151 3/20 0.53
HPGD P15428 3/20 0.53
SMN1; SMN2 Q16637 4/20 0.53
CYP1A2 P05177 2/20 0.53
CYP2C9 P11712 2/20 0.53
CYP2C19 P33261 2/20 0.53
GAA P10253 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6154791 0.91 HDAC6 (0.54) HDAC6RARARARBRARGNPC1
SCHEMBL28587303 0.82 HDAC6 (0.62) HDAC6NPC1MEN1KMT2ADHODH
SCHEMBL15515850 0.79 KDM4E (0.60) RARARARBRARGNPC1MEN1
SCHEMBL491414 0.79 MEN1 (0.64) RARARARBRARGNPC1MEN1
SCHEMBL9176722 0.78 SMN1; SMN2 (0.72) NPC1MEN1KMT2AGBA1MAPT
SCHEMBL28574866 0.77 HDAC6 (0.61) HDAC6NPC1MEN1KMT2AMAPT
SCHEMBL24233043 0.77 KMT2A (0.71) MEN1KMT2AMAPTLMNAPOLB
SCHEMBL2423069 0.77 KDM4E (0.74) NPC1LMNARAB9AHPGDSMN1; SMN2
SCHEMBL2179717 0.76 TRPM8 (0.58) RARARARBRARGNPC1MEN1
SCHEMBL5557794 0.76 HDAC6 (0.52) HDAC6NPC1MEN1KMT2ARXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112981436-B Method for synthesizing 2-amino-1, 3, 4-thiadiazole derivative through electrochemical oxidation 昆明学院 2022-02-01 CN claimed
CN-112981436-A Method for synthesizing 2-amino-1, 3, 4-thiadiazole derivative through electrochemical oxidation 昆明学院 2021-06-18 CN claimed
CN-112981436-B Method for synthesizing 2-amino-1, 3, 4-thiadiazole derivative through electrochemical oxidation 昆明学院 2022-02-01 CN disclosed
CN-112981436-A Method for synthesizing 2-amino-1, 3, 4-thiadiazole derivative through electrochemical oxidation 昆明学院 2021-06-18 CN disclosed