Choline

Choline

SCHEMBL28574563

C=C(C)C(=O)OOP(=O)(O)O.C[N+](C)(C)CCO

nearest known ligand 0.39

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADORA1ADORA2AADORA2BADORA3GNRHRMPLPDE3APDE3BPDE4APDE4BPDE4CPDE4DPPARASLC5A2

The experimentally established mechanism targets of Choline. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.38
LMNA P02545 1/20 0.38
KMT2A Q03164 1/20 0.38
CYP3A4 P08684 1/20 0.38
SLC5A7 Q9GZV3 1/20 0.38
GALR3 O60755 2/20 0.32
BBOX1 O75936 2/20 0.32
CHRM5 P08912 2/20 0.32
CHRM1 P11229 2/20 0.32
CHRM3 P20309 2/20 0.32
PGR P06401 1/20 0.32
CHRM2 P08172 1/20 0.32
CHRM4 P08173 1/20 0.32
HTR1A P08908 1/20 0.32
CHRNB2 P17787 1/20 0.32
TBXA2R P21731 1/20 0.32
CHRNB4 P30926 1/20 0.32
CHRNA3 P32297 1/20 0.32
CHRNA7 P36544 1/20 0.32
CHRNA4 P43681 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Choline SCHEMBL27883877 0.86 MEN1 (0.34) MEN1LMNAKMT2ACYP3A4SLC5A7
Ethylene Glycol SCHEMBL2336848 0.86 ALDH1A1 (0.38) ALDH1A1TSHR
SCHEMBL908616 0.82 ALDH1A1 (0.44) ALDH1A1TSHR
Choline SCHEMBL28025633 0.80 TSHR (0.36) LMNACYP3A4TSHR
Choline SCHEMBL21587444 0.77 THRB (0.42) MEN1LMNAKMT2ACYP3A4SLC5A7
SCHEMBL28151167 0.76 CHRM5 (0.38) LMNAGALR3CHRM5CHRM1CHRM3
Choline SCHEMBL29084705 0.76 TSHR (0.33) MEN1LMNAKMT2ACYP3A4SLC5A7
Choline SCHEMBL27577904 0.75 BBOX1 (0.43) MEN1LMNAKMT2ACYP3A4SLC5A7
SCHEMBL30877085 0.72 SMN1; SMN2 (0.46) LMNAGALR3CHRM5CHRM1CHRM3
Choline SCHEMBL28428557 0.72 GALR3 (0.40) MEN1LMNAKMT2ACYP3A4SLC5A7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112972428-B Mesoporous silicon-based drug carrier coated by zwitterionic polymer film and preparation method thereof 石河子大学 2022-03-08 CN disclosed
CN-112972428-A Mesoporous silicon-based drug carrier coated by zwitterionic polymer film and preparation method thereof 石河子大学 2021-06-18 CN disclosed