SCHEMBL28575012

SCHEMBL28575012

N#Cc1cc(Cl)c(N=C=O)c(Cl)c1

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
VCAM1 P19320 3/20 0.37
GABRA1 P14867 1/20 0.35
GABRB2 P47870 1/20 0.35
GPR35 Q9HC97 1/20 0.33
FASN P49327 1/20 0.31
TTR P02766 2/20 0.30
ALB P02768 2/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
AR P10275 2/20 0.30
HSD11B1 P28845 1/20 0.30
MRGPRX4 Q96LA9 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28912552 0.87 MAPK1 (0.34) MAPK1TDP1VCAM1GABRA1GABRB2
SCHEMBL4009416 0.79 GABRA1 (0.34) VCAM1GABRA1GABRB2GPR35TTR
SCHEMBL1019709 0.78 MAPK1 (0.45) MAPK1TDP1GABRA1GABRB2MEN1
SCHEMBL5206535 0.76 MAPK1 (0.59) MAPK1TDP1GABRA1GABRB2
SCHEMBL28560711 0.75 VCAM1 (0.32) VCAM1GABRA1GABRB2TTRALB
SCHEMBL28566732 0.75 VCAM1 (0.42) MAPK1TDP1VCAM1ARHSD11B1
SCHEMBL1950823 0.74 MAPK1 (0.42) MAPK1TDP1GABRA1GABRB2
SCHEMBL6330610 0.74 MAPK1 (0.42) MAPK1TDP1GABRA1GABRB2
SCHEMBL11322087 0.74 GABRA1 (0.42) MAPK1TDP1GABRA1GABRB2GPR35
SCHEMBL8641955 0.73 MAPK1 (0.50) MAPK1TDP1GABRA1GABRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113248506-A Substituted aminopurine compounds, compositions thereof, and methods of treatment therewith 西格诺药品有限公司 2021-08-13 CN disclosed
CN-107001372-B Substituted aminopurine compounds, compositions thereof, and methods of treatment therewith 西格诺药品有限公司 2021-04-27 CN disclosed