SCHEMBL28575823

SCHEMBL28575823

CC(C)(C#N)CCOc1ccccc1-c1nccc(C(=O)O)n1

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
XDH P47989 10/20 0.45
PTGER1 P34995 1/20 0.39
IDO1 P14902 1/20 0.37
USP2 O75604 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
TSHR P16473 1/20 0.35
CYP2C19 P33261 1/20 0.35
PPARG P37231 1/20 0.35
MAPT P10636 1/20 0.35
THRB P10828 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28600234 0.82 IDO1 (0.42) XDHIDO1PPARG
SCHEMBL28574651 0.82 XDH (0.47) XDHPTGER1
SCHEMBL28586213 0.81 ALDH1A1 (0.43) XDHPTGER1IDO1PPARG
SCHEMBL28570870 0.80 XDH (0.54) XDHPTGER1IDO1
SCHEMBL28579825 0.79 XDH (0.50) XDHPTGER1USP2TSHRMAPT
SCHEMBL28568681 0.77 PDE5A (0.38) IDO1USP2CYP1A2PPARGMAPT
SCHEMBL28570869 0.76 XDH (0.48) XDHPTGER1USP2CYP1A2CYP3A4
SCHEMBL28914642 0.76 XDH (0.45) XDHPTGER1USP2CYP1A2CYP3A4
SCHEMBL28579824 0.72 XDH (0.46) XDHPTGER1USP2CYP1A2CYP3A4
SCHEMBL28583440 0.72 XDH (0.59) XDHPTGER1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112979559-A 2-phenyl pyrimidine formic acid derivative and preparation method and application thereof 沈阳药科大学 2021-06-18 CN claimed
CN-112979559-A 2-phenyl pyrimidine formic acid derivative and preparation method and application thereof 沈阳药科大学 2021-06-18 CN disclosed