SCHEMBL28577976

SCHEMBL28577976

COC(=O)c1ccc(C(=O)CCCCNC(=O)OC(C)(C)C)cc1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 2/20 0.50
TDP1 Q9NUW8 1/20 0.50
POLB P06746 1/20 0.49
BRD4 O60885 1/20 0.47
CYP3A4 P08684 1/20 0.46
CA1 P00915 7/20 0.45
CA2 P00918 7/20 0.45
CA12 O43570 5/20 0.45
CA9 Q16790 5/20 0.45
MAOA P21397 1/20 0.45
MAOB P27338 1/20 0.45
MEN1 O00255 1/20 0.44
GAA P10253 1/20 0.44
KMT2A Q03164 1/20 0.44
DRD2 P14416 1/20 0.43
KDM4E B2RXH2 1/20 0.43
MAPT P10636 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4085154 0.96 MGLL (0.48) MGLLTDP1POLBBRD4CA1
SCHEMBL30905400 0.86 POLB (0.67) MGLLTDP1POLBBRD4CA1
SCHEMBL10322699 0.86 L3MBTL1 (0.53) TDP1CYP3A4CA1CA2CA12
SCHEMBL16409222 0.84 TDP1 (0.48) TDP1BRD4CYP3A4CA1CA2
SCHEMBL2333929 0.84 CYP4A11 (0.58) MGLLTDP1POLBBRD4CA1
SCHEMBL15856116 0.83 CA12 (0.66) MGLLTDP1POLBCA1CA2
SCHEMBL24350075 0.82 NPC1 (0.54) TDP1POLBCA1CA2CA12
SCHEMBL1760150 0.82 HDAC1 (0.49) TDP1CA1CA2CA12CA9
SCHEMBL21221559 0.82 CYP4A11 (0.57) MGLLTDP1POLBBRD4CA1
SCHEMBL1929771 0.82 SIGMAR1 (0.52) TDP1CYP3A4CA1CA2CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113072521-B ROR gamma t inhibitor and application thereof in medicines 广东东阳光药业股份有限公司 2024-04-05 CN disclosed
CN-113072542-B ROR gamma t inhibitor and preparation method and application thereof 广东东阳光药业股份有限公司 2024-04-05 CN disclosed
CN-113072521-A ROR gamma t inhibitor and application thereof in medicine 广东东阳光药业有限公司 2021-07-06 CN disclosed
CN-113072542-A ROR gamma t inhibitor and preparation method and application thereof 广东东阳光药业有限公司 2021-07-06 CN disclosed