SCHEMBL28579575

SCHEMBL28579575

COC(=O)c1ccccc1NC(=O)c1c[nH]c2ccccc12

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.72
KMT2A Q03164 2/20 0.72
MEN1 O00255 1/20 0.72
NR4A2 P43354 2/20 0.71
CREBBP Q92793 1/20 0.71
TSHR P16473 6/20 0.58
MAPK1 P28482 2/20 0.58
HSD17B10 Q99714 2/20 0.58
GAA P10253 1/20 0.58
MAPT P10636 1/20 0.58
TDP1 Q9NUW8 1/20 0.56
L3MBTL1 Q9Y468 1/20 0.56
CFTR P13569 2/20 0.55
RAB9A P51151 1/20 0.54
CYP1A2 P05177 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C19 P33261 1/20 0.52
PBRM1 Q86U86 1/20 0.51
APOBEC3A P31941 1/20 0.51
APOBEC3G Q9HC16 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28572431 0.85 NR4A2 (0.61) NPC1KMT2AMEN1NR4A2CREBBP
SCHEMBL28577422 0.85 MEN1 (0.65) NPC1KMT2AMEN1NR4A2CREBBP
SCHEMBL1093530 0.84 NR4A2 (1.00) KMT2AMEN1NR4A2CREBBPMAPT
SCHEMBL30031033 0.84 NR4A2 (1.00) KMT2AMEN1NR4A2CREBBPMAPT
SCHEMBL28569094 0.84 NR4A2 (0.63) NPC1KMT2AMEN1NR4A2CREBBP
SCHEMBL21446804 0.83 ALDH1A1 (0.67) NPC1KMT2AMEN1NR4A2CREBBP
Hydrochloric Acid SCHEMBL28254334 0.82 NR4A2 (0.97) KMT2AMEN1NR4A2CREBBPMAPT
SCHEMBL20567854 0.81 NPC1 (0.68) NPC1KMT2AMEN1NR4A2CREBBP
SCHEMBL27075304 0.81 NPC1 (0.68) NPC1KMT2AMEN1NR4A2CREBBP
SCHEMBL21438794 0.80 NR4A2 (0.79) NPC1KMT2AMEN1NR4A2CREBBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113004188-B Indole derivative, preparation method and application 沈阳药科大学 2022-09-20 CN disclosed
CN-113004188-A Indole derivative, preparation method and application 沈阳药科大学 2021-06-22 CN disclosed