SCHEMBL28580229

SCHEMBL28580229

CNS(=O)(=O)N1CCC(C(F)(F)F)CC1

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 6/20 0.35
CNR2 P34972 3/20 0.35
HSD11B1 P28845 1/20 0.33
JAK2 O60674 1/20 0.33
JAK1 P23458 1/20 0.33
TYK2 P29597 1/20 0.33
JAK3 P52333 1/20 0.33
GAA P10253 1/20 0.33
KCNT1 Q5JUK3 2/20 0.32
POLB P06746 1/20 0.32
CCND1 P24385 2/20 0.31
CCNE1 P24864 2/20 0.31
CDK2 P24941 2/20 0.31
CDK6 Q00534 2/20 0.31
ACLY P53396 1/20 0.31
HCRTR2 O43614 1/20 0.31
SCN9A Q15858 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26470386 0.82 ACLY (0.42) HSD11B1CCND1CCNE1CDK2CDK6
SCHEMBL2104714 0.78 TP53 (0.44) HSD11B1
SCHEMBL25279069 0.76 TP53 (0.38) CNR1CNR2GAAKCNT1ACLY
SCHEMBL14971519 0.75 MEN1 (0.44) POLB
SCHEMBL16825250 0.75 POLB (0.38) CNR1CNR2HSD11B1JAK2JAK1
SCHEMBL1822000 0.75 CA1 (0.42) CNR1CNR2HSD11B1JAK2JAK1
SCHEMBL18711984 0.74 HSD11B1 (0.36) HSD11B1JAK2JAK1TYK2JAK3
SCHEMBL12765367 0.74 MAPK1 (0.40) HSD11B1GAACCND1CCNE1CDK2
SCHEMBL2424959 0.74 CCNE1 (0.33) CCND1CCNE1CDK2CDK6
SCHEMBL2104712 0.74 HSD11B1 (0.35) CNR1CNR2HSD11B1JAK2JAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112830893-A ROR gamma inhibitor, preparation method and medical application thereof 成都倍特药业股份有限公司 2021-05-25 CN disclosed