SCHEMBL28587714

SCHEMBL28587714

NNC(=O)c1ccc(CCS(N)(=O)=O)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 5/20 0.58
CA2 P00918 5/20 0.58
CA9 Q16790 2/20 0.58
RECQL P46063 1/20 0.55
CA12 O43570 1/20 0.51
MPO P05164 2/20 0.50
CYP3A4 P08684 2/20 0.50
KDM5A P29375 1/20 0.50
BLM P54132 1/20 0.50
GFER P55789 1/20 0.50
PMP22 Q01453 1/20 0.50
HIF1A Q16665 1/20 0.50
MAPT P10636 3/20 0.48
ALDH1A1 P00352 3/20 0.48
KDM4E B2RXH2 2/20 0.48
OGG1 O15527 1/20 0.48
LMNA P02545 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
HDAC1 Q13547 2/20 0.44
HDAC8 Q9BY41 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6608511 0.81 RECQL (0.58) CA1CA2CA9RECQLCA12
SCHEMBL691846 0.81 CA1 (0.61) CA1CA2CA9CA12MPO
SCHEMBL28583909 0.76 HDAC1 (0.72) MPOCYP3A4KDM5ABLMGFER
SCHEMBL2678949 0.76 MPO (0.80) CA1CA2CA9RECQLMPO
SCHEMBL11217374 0.76 PLK1 (0.72) CA1CA2MPOCYP3A4KDM5A
SCHEMBL343630 0.76 MPO (0.80) CA1CA2CA9RECQLMPO
SCHEMBL11139882 0.74 MPO (0.64) CA1CA2CA9MPOCYP3A4
SCHEMBL2836138 0.74 CYP3A4 (0.53) CA1CA2CA9MPOCYP3A4
SCHEMBL28188923 0.73 MPO (0.76) CA1CA2CA9RECQLMPO
SCHEMBL4616920 0.73 CA2 (1.00) CA1CA2CA9CA12KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107922362-B 1,3, 4-oxadiazole sulfonamide derivative compounds as histone deacetylase 6 inhibitors and pharmaceutical compositions containing the same 株式会社钟根堂 2021-06-15 CN disclosed