SCHEMBL28587883

SCHEMBL28587883

Nc1cc(-c2ccc(F)c(F)c2)[nH]n1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.62
KMT2A Q03164 2/20 0.62
MKNK1 Q9BUB5 1/20 0.62
MKNK2 Q9HBH9 1/20 0.62
MEN1 O00255 1/20 0.62
USP2 O75604 1/20 0.62
SMN1; SMN2 Q16637 1/20 0.58
NOTUM Q6P988 1/20 0.53
MITF O75030 1/20 0.53
TP53 P04637 1/20 0.53
DYRK1A Q13627 1/20 0.53
LTA4H P09960 1/20 0.53
LMNA P02545 1/20 0.50
NPC1 O15118 1/20 0.50
MAPT P10636 1/20 0.50
RAB9A P51151 1/20 0.50
GFER P55789 1/20 0.50
PDPK1 O15530 1/20 0.42
HSD17B10 Q99714 2/20 0.41
IDO1 P14902 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30512083 1.00 ALDH1A1 (0.62) ALDH1A1KMT2AMKNK1MKNK2MEN1
SCHEMBL1702207 0.81 ALDH1A1 (0.67) ALDH1A1KMT2AMKNK1MKNK2MEN1
SCHEMBL30512080 0.80 DYRK1A (0.60) ALDH1A1KMT2AMKNK1MKNK2MEN1
SCHEMBL28579218 0.80 DYRK1A (0.60) ALDH1A1KMT2AMKNK1MKNK2MEN1
SCHEMBL29004199 0.78 NOTUM (0.53) ALDH1A1KMT2AMKNK1MKNK2MEN1
SCHEMBL13815700 0.77 KMT2A (1.00) ALDH1A1KMT2AMKNK1MKNK2MEN1
SCHEMBL5630086 0.77 MKNK1 (1.00) ALDH1A1KMT2AMKNK1MKNK2MEN1
SCHEMBL1853364 0.76 LMNA (0.56) ALDH1A1KMT2AMKNK1MKNK2MEN1
SCHEMBL28573902 0.76 ALDH1A1 (0.71) ALDH1A1KMT2AMKNK1MKNK2MEN1
SCHEMBL6252242 0.74 MKNK1 (0.68) ALDH1A1KMT2AMKNK1MKNK2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112876482-B Polysubstituted heterocyclic derivative, preparation method and medical application thereof 中国药科大学 2023-07-28 CN disclosed
CN-112876482-A Polysubstituted heterocyclic derivative, preparation method and medical application thereof 中国药科大学 2021-06-01 CN disclosed