SCHEMBL28591998

SCHEMBL28591998

FC(F)(F)c1ccc(-n2nc(C(F)(F)F)[c]c2Cl)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRAF P15056 2/20 0.40
ATM Q13315 1/20 0.40
MAPT P10636 1/20 0.36
RAB9A P51151 1/20 0.36
CTDSP1 Q9GZU7 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
NPBWR1 P48145 2/20 0.36
PTGS2 P35354 3/20 0.36
PTGS1 P23219 1/20 0.36
HIF1A Q16665 1/20 0.35
XDH P47989 1/20 0.35
CYP2C9 P11712 2/20 0.35
SRC P12931 1/20 0.35
KDR P35968 1/20 0.35
KDM4E B2RXH2 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
MCHR1 Q99705 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
PDPK1 O15530 1/20 0.35
SCN9A Q15858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28595989 0.88 PTGS2 (0.46) MAPTL3MBTL1PTGS2PTGS1HIF1A
SCHEMBL28581887 0.87 PTGS2 (0.36) BRAFATMPTGS2PTGS1SRC
SCHEMBL28586026 0.85 PTGS2 (0.36) MAPTRAB9APTGS2PTGS1KDM4E
SCHEMBL4459050 0.85 PTGS1 (0.41) BRAFMAPTRAB9APTGS2PTGS1
SCHEMBL8352171 0.66 MAPT (0.44) BRAFMAPTRAB9ACTDSP1L3MBTL1
SCHEMBL2064542 0.65
SCHEMBL15332005 0.64 BRAF (0.43) BRAFATMMAPTRAB9ACTDSP1
SCHEMBL19120598 0.63 NPBWR1 (0.49) BRAFATMMAPTRAB9ACTDSP1
SCHEMBL19120335 0.63 HIF1A (0.44) BRAFATMMAPTRAB9ACTDSP1
SCHEMBL16927650 0.63 XDH (0.44) BRAFATMMAPTRAB9ACTDSP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108864075-B Isothiazole bithiazole derivative and preparation method and application thereof 南开大学 2021-06-01 CN claimed