SCHEMBL28596201

SCHEMBL28596201

CCn1c(-c2ccc(C(=O)OC)cc2)nc2ccccc21

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 5/20 0.71
TBXA2R P21731 5/20 0.71
PTGER4 P35408 4/20 0.67
KDM4E B2RXH2 8/20 0.61
ALDH1A1 P00352 5/20 0.61
HPGD P15428 2/20 0.61
SMN1; SMN2 Q16637 3/20 0.59
NPSR1 Q6W5P4 2/20 0.59
NPC1 O15118 2/20 0.59
MAPT P10636 2/20 0.59
RAB9A P51151 2/20 0.59
HTT P42858 2/20 0.59
MEN1 O00255 1/20 0.59
CYP1A2 P05177 1/20 0.59
CYP3A4 P08684 1/20 0.59
CYP2C9 P11712 1/20 0.59
CYP2C19 P33261 1/20 0.59
GFER P55789 1/20 0.59
KMT2A Q03164 1/20 0.59
LMNA P02545 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28600078 0.90 DRD2 (0.69) DRD2TBXA2RPTGER4KDM4EALDH1A1
SCHEMBL28597103 0.88 DRD2 (0.66) DRD2TBXA2RPTGER4KDM4EALDH1A1
SCHEMBL28610296 0.86 PTGER4 (0.67) DRD2TBXA2RPTGER4KDM4EALDH1A1
SCHEMBL31472968 0.85 HDAC6 (0.62) DRD2TBXA2RPTGER4KDM4EALDH1A1
SCHEMBL2879379 0.84 DRD2 (0.85) DRD2TBXA2RKDM4EALDH1A1HPGD
SCHEMBL3497345 0.83 DRD2 (0.62) DRD2TBXA2RKDM4EALDH1A1HPGD
SCHEMBL17938355 0.81 PTGER4 (1.00) PTGER4
SCHEMBL17938347 0.80 PTGER4 (0.86) PTGER4
SCHEMBL10080422 0.80 KDM4E (0.80) DRD2KDM4EALDH1A1HPGDSMN1; SMN2
SCHEMBL11313561 0.79 KDM4E (0.73) KDM4EALDH1A1HPGDSMN1; SMN2NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113166073-A Benzoheterocyclic compounds and compositions for preventing or treating cancer diseases containing the same as active ingredient 启明大学校产学协力团 2021-07-23 CN disclosed