SCHEMBL28596221

SCHEMBL28596221

Cc1c[c]c(-n2cncn2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
CYP2A6 P11509 1/20 0.37
CYP1A2 P05177 3/20 0.35
CYP2C19 P33261 3/20 0.35
CYP2C9 P11712 2/20 0.35
CYP2D6 P10635 2/20 0.35
ADORA2A P29274 1/20 0.34
ADORA1 P30542 1/20 0.34
CYP3A4 P08684 2/20 0.33
POLB P06746 2/20 0.33
HSP90AA1 P07900 2/20 0.32
MAPT P10636 1/20 0.32
HTT P42858 1/20 0.32
KMT2A Q03164 1/20 0.31
PDE4B Q07343 1/20 0.31
FBP1 P09467 1/20 0.30
KCNJ5 P48544 1/20 0.30
KCNJ3 P48549 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28596244 0.80 KDM4E (0.38) SMN1; SMN2KDM4EALDH1A1CYP2A6CYP1A2
SCHEMBL1196464 0.80 CYP19A1 (0.39) SMN1; SMN2KDM4EALDH1A1CYP2A6POLB
SCHEMBL28589922 0.80 MAOB (0.42) SMN1; SMN2KDM4EALDH1A1CYP2A6CYP1A2
SCHEMBL28609555 0.76 ALDH1A1 (0.38) SMN1; SMN2KDM4EALDH1A1CYP2A6CYP1A2
SCHEMBL10515945 0.75 CYP2A6 (0.39) SMN1; SMN2KDM4EALDH1A1CYP2A6CYP1A2
SCHEMBL4616384 0.74 CYP1A2 (0.40) SMN1; SMN2KDM4EALDH1A1CYP1A2CYP2C19
SCHEMBL28597901 0.73 SMN1; SMN2 (0.36) SMN1; SMN2KDM4EALDH1A1CYP2A6CYP1A2
SCHEMBL82347 0.72 SMN1; SMN2 (0.60) SMN1; SMN2KDM4EALDH1A1CYP2A6CYP1A2
SCHEMBL586172 0.72 CYP2A6 (0.42) SMN1; SMN2KDM4EALDH1A1CYP2A6CYP1A2
SCHEMBL17007372 0.70 NOTUM (0.39) KDM4EALDH1A1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113164458-A Monoacylglycerol lipase modulators 詹森药业有限公司 2021-07-23 CN claimed
CN-113164458-A Monoacylglycerol lipase modulators 詹森药业有限公司 2021-07-23 CN disclosed