SCHEMBL28599998

SCHEMBL28599998

CC(C)Cn1cc(C#N)c2ccc(N)cc21

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
XDH P47989 2/20 0.48
STAT3 P40763 1/20 0.40
PFKFB1 P16118 6/20 0.39
PFKFB3 Q16875 6/20 0.39
PFKFB2 O60825 5/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
POLB P06746 1/20 0.39
ALDH1A1 P00352 2/20 0.38
MEN1 O00255 1/20 0.38
TSHR P16473 1/20 0.38
KMT2A Q03164 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
NR3C1 P04150 1/20 0.38
PGR P06401 1/20 0.38
NR3C2 P08235 1/20 0.38
CYP3A4 P08684 1/20 0.38
MAPT P10636 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28597332 0.89 XDH (0.54) XDHSTAT3PFKFB1PFKFB3PFKFB2
SCHEMBL28592975 0.78 XDH (0.45) XDHALDH1A1NR3C1PGRNR3C2
SCHEMBL28592963 0.78 XDH (0.44) XDHPFKFB1PFKFB3PFKFB2SMN1; SMN2
SCHEMBL28601590 0.77 STAT3 (0.46) XDHSTAT3SMN1; SMN2POLBALDH1A1
SCHEMBL28608931 0.77 XDH (0.45) XDHSTAT3SMN1; SMN2POLBALDH1A1
SCHEMBL28918220 0.76 XDH (0.49) XDHSTAT3SMN1; SMN2POLBALDH1A1
SCHEMBL2850331 0.75 IMPDH2 (0.59) ALDH1A1
Hydrochloric Acid SCHEMBL28606116 0.74 XDH (0.54) XDHSTAT3SMN1; SMN2POLBMAPT
SCHEMBL22803875 0.73 POLB (0.37) STAT3SMN1; SMN2POLBALDH1A1TSHR
SCHEMBL24143651 0.70 NR1D1 (0.51)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113173918-B N-indole-1, 6-dihydropyrimidine-4-carboxamide derivative and preparation method and application thereof 沈阳药科大学 2022-04-05 CN disclosed
CN-113173918-A N-indole-1, 6-dihydropyrimidine-4-carboxamide derivative and preparation method and application thereof 沈阳药科大学 2021-07-27 CN disclosed