SCHEMBL2860019

SCHEMBL2860019

Cc1ccc(Nc2nc(-c3cccc(C(C)C)c3)nc3c2cnn3C)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 7/20 0.58
HTR2C P28335 3/20 0.50
HAVCR2 Q8TDQ0 1/20 0.49
GGPS1 O95749 1/20 0.48
BCDIN3D Q7Z5W3 3/20 0.46
BTK Q06187 1/20 0.46
MAPT P10636 3/20 0.45
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
KDM4E B2RXH2 2/20 0.45
MAPK1 P28482 2/20 0.45
ALDH1A1 P00352 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
LMNA P02545 1/20 0.45
TP53 P04637 1/20 0.45
ABCG2 Q9UNQ0 1/20 0.45
HCRTR1 O43613 1/20 0.44
CYP1A2 P05177 1/20 0.44
POLB P06746 1/20 0.44
HSP90AA1 P07900 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2870134 0.87 HTR2C (0.53) PIK3CAHTR2CHAVCR2MAPTMEN1
SCHEMBL2875609 0.80 HTR2C (0.67) PIK3CAHTR2CHAVCR2BCDIN3DMAPT
SCHEMBL31194469 0.74 PDE5A (0.61) PIK3CAHTR2CBCDIN3DMAPTMEN1
SCHEMBL3184819 0.74 PIK3CA (0.54) PIK3CAHTR2CGGPS1BCDIN3DBTK
SCHEMBL2806838 0.73 PIK3CA (0.61) PIK3CAGGPS1BCDIN3DBTKMAPT
SCHEMBL2804510 0.73 NPC1 (0.47) PIK3CAHTR2CHAVCR2GGPS1MAPT
SCHEMBL3174574 0.73 PIK3CA (0.64) PIK3CAHTR2CGGPS1BCDIN3DBTK
SCHEMBL13087256 0.72 GAA (0.78) HTR2CHAVCR2MAPTMEN1KMT2A
SCHEMBL3175599 0.71 PIK3CA (0.62) PIK3CAHTR2CBCDIN3DBTKMAPT
SCHEMBL3181720 0.70 PIK3CA (0.63) PIK3CAHTR2CGGPS1BCDIN3DBTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010118367-A2 ANTIVIRAL PYRIMIDINES PROGENICS PHARMACEUTICALS, INC. (US) 2010-10-14 WO disclosed