SCHEMBL28600460

SCHEMBL28600460

O=C(O)Nc1ccccc1-c1ccccc1C1CCNCC1

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 4/20 0.50
HTR2C P28335 6/20 0.47
CHRM1 P11229 3/20 0.47
CHRM2 P08172 2/20 0.47
P2RY14 Q15391 1/20 0.43
HTR1A P08908 1/20 0.42
SLC6A2 P23975 1/20 0.42
SLC6A4 P31645 1/20 0.42
SLC6A3 Q01959 1/20 0.42
SLC18A3 Q16572 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
JAK3 P52333 1/20 0.41
ALDH1A1 P00352 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8553355 0.88 HTR2C (0.53) CHRM3HTR2CHTR1ASLC6A2SLC6A4
SCHEMBL28666071 0.78 CHRM3 (0.48) CHRM3HTR2CCHRM1CHRM2
SCHEMBL27561971 0.75 HTR2C (0.51) CHRM3HTR2CHTR1ASLC6A2SLC6A4
SCHEMBL83107 0.74 CETP (0.48) CHRM3HTR2C
Hydrochloric Acid SCHEMBL7669676 0.74 HTR2C (0.53) HTR2CHTR1ASLC6A2SLC6A4SLC6A3
SCHEMBL2060591 0.74 HSD17B10 (0.43) CHRM3ALDH1A1
SCHEMBL5599211 0.73 HSD17B10 (0.51) ALDH1A1
SCHEMBL3121349 0.73 HTR2C (0.56) HTR2CHTR1ASLC6A2SLC6A4SLC6A3
SCHEMBL7676995 0.72 HTR2C (0.53) CHRM3HTR2CCHRM1CHRM2HTR1A
SCHEMBL4639850 0.72 P2RY14 (0.56) P2RY14SLC18A3SIGMAR1JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113121412-A Preparation method of lefenacin intermediate 扬州中宝药业股份有限公司 2021-07-16 CN disclosed