SCHEMBL28601844

SCHEMBL28601844

CC(C)(C)C(OC(N)=O)c1ccc(CN)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LOXL2 Q9Y4K0 3/20 0.41
BACE1 P56817 1/20 0.37
NOS3 P29474 2/20 0.36
NOS1 P29475 2/20 0.36
NOS2 P35228 2/20 0.36
EPHX1 P07099 2/20 0.36
KDM4E B2RXH2 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
PLG P00747 3/20 0.35
KLK1 P06870 2/20 0.35
KLK6 Q92876 2/20 0.35
TPSAB1 Q15661 5/20 0.35
HDAC3 O15379 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
NCOR2 Q9Y618 1/20 0.35
ABAT P80404 1/20 0.34
F10 P00742 1/20 0.34
PRSS1 P07477 2/20 0.33
TPSD1 Q9BZJ3 1/20 0.33
TPSG1 Q9NRR2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29007663 0.86 EPHX1 (0.35) EPHX1
SCHEMBL5026454 0.81 PARP10 (0.34) KDM4ESMN1; SMN2
SCHEMBL31348907 0.80 ALOX5 (0.44) EPHX1SMN1; SMN2
SCHEMBL29156721 0.79 NPSR1 (0.47)
SCHEMBL31267216 0.77 TDP1 (0.33)
SCHEMBL5026419 0.73
SCHEMBL28552109 0.73 MAPK1 (0.50) SMN1; SMN2
SCHEMBL29243385 0.71 ALOX5 (0.50) KDM4E
SCHEMBL28540156 0.71 F11 (0.45) F10PRSS1
SCHEMBL25339719 0.71 SLC6A3 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113004286-A Tricyclic compounds as plasma kallikrein inhibitors and uses thereof 成都康弘药业集团股份有限公司 2021-06-22 CN disclosed