SCHEMBL28604392

SCHEMBL28604392

CCOS(=O)(=O)c1ccc(C)cc1C1(O)CCC(NC(=O)OC(C)(C)C)CC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.38
MAOB P27338 2/20 0.36
KDM1A O60341 1/20 0.36
MAPT P10636 1/20 0.36
DRD2 P14416 4/20 0.35
CTSL P07711 1/20 0.35
CTSB P07858 1/20 0.35
CTSS P25774 1/20 0.35
CTSK P43235 1/20 0.35
KAT6A Q92794 1/20 0.35
KAT5 Q92993 1/20 0.35
KMT2A Q03164 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
ALDH1A1 P00352 1/20 0.35
BRD4 O60885 2/20 0.35
GAA P10253 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
KCNA3 P22001 1/20 0.34
PKM P14618 1/20 0.34
RORC P51449 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28587573 0.89 EPHX2 (0.37) EPHX2MAOBKDM1AMAPTDRD2
SCHEMBL28479502 0.81 JAK2 (0.41) EPHX2MAOBKDM1AMAPTDRD2
SCHEMBL28576703 0.81 L3MBTL1 (0.35) MAPTDRD2KAT6AKMT2AL3MBTL1
SCHEMBL28476786 0.79 KMT2A (0.40) EPHX2MAOBKDM1AMAPTDRD2
SCHEMBL28789549 0.76 CYP3A4 (0.37) MAPTDRD2KMT2AL3MBTL1ALDH1A1
SCHEMBL28591857 0.75 BRD4 (0.37) EPHX2MAOBKDM1ADRD2CTSL
SCHEMBL28421464 0.73 CYP1A2 (0.48) MAPTKMT2AL3MBTL1ALDH1A1GAA
SCHEMBL30890924 0.72 EPHX2 (0.38) EPHX2MAOBKDM1AMAPTDRD2
SCHEMBL28341524 0.72 EPHX2 (0.48) EPHX2MAOBKDM1AMAPTDRD2
SCHEMBL28597610 0.71 RORC (0.38) EPHX2MAOBKDM1ADRD2KAT6A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112778183-B Nitrogen-containing ring derivative regulator, preparation method and application thereof 江苏豪森药业集团有限公司 2024-05-10 CN disclosed
CN-113166135-A Benzothiophene derivative modulators, methods of making, and uses thereof 上海翰森生物医药科技有限公司 2021-07-23 CN disclosed
CN-112778183-A Nitrogen-containing ring derivative regulator, preparation method and application thereof 江苏豪森药业集团有限公司 2021-05-11 CN disclosed