SCHEMBL28604758

SCHEMBL28604758

CC(C)[Si](C#CC(=O)Cc1ccc(F)cc1)(C(C)C)C(C)C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.44
TDP1 Q9NUW8 2/20 0.42
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
POLB P06746 1/20 0.40
APEX1 P27695 1/20 0.40
LMNA P02545 5/20 0.39
KDM4E B2RXH2 3/20 0.39
MAPT P10636 2/20 0.39
TP53 P04637 1/20 0.39
ALOX15 P16050 1/20 0.39
MAPK1 P28482 1/20 0.39
HSD17B10 Q99714 1/20 0.39
GAA P10253 2/20 0.39
KMT2A Q03164 2/20 0.39
HPGD P15428 1/20 0.39
ALDH1A1 P00352 1/20 0.38
CTBP2 P56545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28920257 0.86 HPGD (0.44) TDP1LMNAGAAKMT2AHPGD
SCHEMBL28605788 0.84 TSHR (0.45) POLBKDM4EMAPTKMT2AALDH1A1
SCHEMBL28607997 0.82 ANPEP (0.40) CYP2D6CYP2C9CYP2C19MAPTALOX15
SCHEMBL28610799 0.82 HTT (0.47) HTTTDP1CYP3A4KDM4ETP53
SCHEMBL28608951 0.82 ACACB (0.40) LMNAMAPTTP53ALDH1A1SMN1; SMN2
SCHEMBL28613558 0.80 KMT2A (0.45) HTTCYP2C19POLBLMNAMAPT
SCHEMBL28609788 0.77 L3MBTL1 (0.44) KMT2A
SCHEMBL28608905 0.75 CTBP2 (0.44) POLBALDH1A1CTBP2NPC1
SCHEMBL28612288 0.74 PTGES (0.40)
SCHEMBL28623769 0.74 PIK3CA (0.45) MAPTKMT2AHPGDALDH1A1CTBP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109942612-B Diyne enamine compound and preparation method and application thereof 北京大学深圳研究生院 2021-08-20 CN disclosed