SCHEMBL28610799

SCHEMBL28610799

COc1ccc(CC(=O)C#C[Si](C(C)C)(C(C)C)C(C)C)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.47
USP2 O75604 1/20 0.44
TP53 P04637 1/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
LDHA P00338 1/20 0.44
PKM P14618 2/20 0.43
CTBP2 P56545 1/20 0.43
ALDH1A1 P00352 3/20 0.43
KLK7 P49862 1/20 0.43
KMT2A Q03164 2/20 0.43
ATM Q13315 2/20 0.43
TDP1 Q9NUW8 2/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
MEN1 O00255 1/20 0.43
NPC1 O15118 1/20 0.43
CYP3A4 P08684 1/20 0.43
HPGD P15428 1/20 0.43
RAB9A P51151 1/20 0.43
KDM4E B2RXH2 1/20 0.42
CDK5 Q00535 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28605790 0.83 CTBP2 (0.48) HTTSMN1; SMN2CTBP2ALDH1A1KMT2A
SCHEMBL28920257 0.83 HPGD (0.44) SMN1; SMN2CTBP2KMT2ATDP1L3MBTL1
SCHEMBL28604758 0.82 HTT (0.44) HTTTP53SMN1; SMN2CTBP2ALDH1A1
SCHEMBL28605788 0.81 TSHR (0.45) SMN1; SMN2ALDH1A1KMT2AL3MBTL1MEN1
SCHEMBL28608951 0.79 ACACB (0.40) TP53SMN1; SMN2ALDH1A1NPC1RAB9A
SCHEMBL28613558 0.77 KMT2A (0.45) HTTPKMALDH1A1KMT2AMEN1
SCHEMBL28609788 0.77 L3MBTL1 (0.44) KMT2AL3MBTL1MEN1
SCHEMBL10445335 0.73 HTT (0.58) HTTUSP2TP53SMN1; SMN2LDHA
SCHEMBL28608905 0.72 CTBP2 (0.44) PKMCTBP2ALDH1A1L3MBTL1NPC1
SCHEMBL28824698 0.72 NPC1 (0.57) HTTUSP2TP53SMN1; SMN2CTBP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109942612-B Diyne enamine compound and preparation method and application thereof 北京大学深圳研究生院 2021-08-20 CN disclosed