SCHEMBL2860487

SCHEMBL2860487

Cn1nc(-c2ccccc2)cc1NC(=O)Oc1cnn(-c2ccc(OC(F)(F)F)cc2)c1C(F)(F)F

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 1/20 0.42
GRM5 P41594 1/20 0.41
MAPT P10636 6/20 0.41
RAB9A P51151 1/20 0.41
XBP1 P17861 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
POLB P06746 2/20 0.39
EPHX2 P34913 1/20 0.39
PTGS2 P35354 1/20 0.39
HTR2A P28223 1/20 0.39
P2RY1 P47900 1/20 0.38
CDK1 P06493 1/20 0.38
CDK4 P11802 1/20 0.38
CCNB1 P14635 1/20 0.38
CCNA2 P20248 1/20 0.38
CCND1 P24385 1/20 0.38
CDK2 P24941 1/20 0.38
CDK7 P50613 1/20 0.38
CCNH P51946 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2858621 0.90 MAPT (0.48) NTRK1GRM5MAPTRAB9AXBP1
SCHEMBL2849954 0.87 MAPT (0.46) NTRK1GRM5MAPTRAB9AXBP1
SCHEMBL2856128 0.85 GRM5 (0.46) NTRK1GRM5MAPTRAB9AXBP1
SCHEMBL2858606 0.79 P2RY1 (0.47) MAPTPOLBEPHX2P2RY1
SCHEMBL2856867 0.77 NPC1 (0.53) MAPTRAB9AHTR2AP2RY1
SCHEMBL2861646 0.77 NPC1 (0.42) MAPTRAB9ANPSR1HTR2AP2RY1
SCHEMBL2853031 0.76 MAPT (0.41) MAPTNPSR1POLBP2RY1
SCHEMBL2855275 0.76 MAPT (0.45) MAPTRAB9AEPHX2P2RY1
SCHEMBL2861443 0.75 MEN1 (0.47) NTRK1MAPTNPSR1P2RY1
SCHEMBL2856517 0.75 MAPT (0.42) MAPTPOLBP2RY1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed