SCHEMBL286072

SCHEMBL286072

C1CCN(C2CCCC[N]2)CC1

nearest known ligand 0.35

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 3/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
LMNA P02545 1/20 0.32
HTR6 P50406 1/20 0.30
CHRM5 P08912 1/20 0.30
ADRA2C P18825 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8640560 1.00 CYP2D6 (0.32) CYP2D6MEN1KMT2ALMNAHTR6
SCHEMBL3558101 1.00 CYP2D6 (0.32) CYP2D6MEN1KMT2ALMNAHTR6
SCHEMBL6050828 1.00 CYP2D6 (0.32) CYP2D6MEN1KMT2ALMNAHTR6
SCHEMBL10891279 1.00 CYP2D6 (0.32) CYP2D6MEN1KMT2ALMNAHTR6
SCHEMBL2569149 1.00 CYP2D6 (0.32) CYP2D6MEN1KMT2ALMNAHTR6
SCHEMBL8640554 1.00 CYP2D6 (0.32) CYP2D6MEN1KMT2ALMNAHTR6
SCHEMBL2229452 1.00 CYP2D6 (0.32) CYP2D6MEN1KMT2ALMNAHTR6
SCHEMBL3658217 1.00 CYP2D6 (0.32) CYP2D6MEN1KMT2ALMNAHTR6
SCHEMBL4712511 1.00 CYP2D6 (0.32) CYP2D6MEN1KMT2ALMNAHTR6
SCHEMBL157427 0.98 CYP2D6 (0.33) CYP2D6MEN1KMT2ALMNAHTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 217 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118146224-A Nitrogen-containing tricyclic derivative and application thereof in medicine 西藏海思科制药有限公司 2024-06-07 CN claimed
CN-117720517-A AR inhibitor, composition thereof and pharmaceutical application thereof 西藏海思科制药有限公司 2024-03-19 CN claimed
WO-2024012570-A1 NITROGEN-CONTAINING HETEROCYCLIC DERIVATIVE, AND COMPOSITION AND PHARMACEUTICAL USE THEREOF 西藏海思科制药有限公司 2024-01-18 WO claimed
WO-2023232133-A1 COMPOUND FOR INHIBITING OR DEGRADING BCL6 AND USE THEREOF IN PHARMACEUTICS 西藏海思科制药有限公司 2023-12-07 WO claimed
WO-2023208165-A1 NITROGEN-CONTAINING HETEROCYCLIC DERIVATIVE, AND COMPOSITION AND PHARMACEUTICAL APPLICATION THEREOF 四川海思科制药有限公司 2023-11-02 WO claimed
CN-116969921-A Compound for inhibiting or degrading HPK1 kinase and application thereof in medicine 四川海思科制药有限公司 2023-10-31 CN claimed
CN-116947877-A Benzimidazole derivative and application thereof in medicine 四川海思科制药有限公司 2023-10-27 CN claimed
EP-3873599-B1 PYRIDINYL SULFONAMIDE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS AND USES THEREOF BOEHRINGER INGELHEIM INT (DE) 2023-09-27 EP claimed
US-11639352-B2 Benzothiazole compounds for the treatment of autoimmune diseases HOFFMAN-LA ROCHE INC. (US) 2023-05-02 US claimed
CN-114920746-A BTK (BTK inhibitory or degrading agent) and application thereof in medicine 四川海思科制药有限公司 2022-08-19 CN claimed
WO-2005089747-A1 NOVEL AZABICYCLIC DERIVATIVES, PREPARATION METHOD THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME LES LABORATOIRES SERVIER (FR) 2005-09-29 WO claimed
US-6908929-B2 Phenyl-substituted imidazopyridines ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2005-06-21 US claimed
US-20050090523-A1 2-(substituted phenyl)imidazo[1,2-a]pyridine compounds; use to treat disorders mediated by the histamine H3 receptor such as sleep disorders, attention deficit hyperactivity disorder, or Alzheimer's disease; 2-[4-[3-(Piperidino)propylamino]phenyl]-8-methylimidazo[1,2-a]pyridine for example BREITENBUCHER J G (US) 2005-04-28 US claimed
US-20050085502-A1 Phenyl-substituted imidazopyridines BREITENBUCHER J G (US) 2005-04-21 US claimed
US-6734306-B2 USEFUL IN THE TREATMENT OF INFLAMMATION, ASTHMA, ALLERGIC RHINITIS, PAIN OR THE LIKE PFIZER, INC. 2004-05-11 US claimed
EP-1268478-A2 PHENYL-SUBSTITUTED IMIDAZOPYRIDINES Ortho McNeil Pharmaceutical, Inc. (US) 2003-01-02 EP claimed
US-20020128271-A1 N-benzenesulfonyl l-proline compounds as bradykinin antagonists PFIZER INC. 2002-09-12 US claimed
EP-1213289-A1 N-benzenesulfonyl L-proline compounds as bradykinin antagonists PFIZER INC. (US) 2002-06-12 EP claimed
US-20020006934-A1 Phenyl-substituted imidazopyridines ORTHO MCNEIL PHARMACEUTICAL, INC. 2002-01-17 US claimed
WO-2001074815-A2 PHENYL-SUBSTITUTED IMIDAZOPYRIDINES ORTHO MCNEIL PHARMACEUTICAL, INC. (US) 2001-10-11 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050085502-A1 Phenyl-substituted imidazopyridines AADAC, DPP4, DPP3 CYP2D6 46/4885MEN1 4485/4885KMT2A 2545/4885
US-20020128271-A1 N-benzenesulfonyl l-proline compounds as bradykinin antagonists BDKRB1, HRH2, BDKRB2 CYP2D6 2011/4885MEN1 3988/4885KMT2A 2975/4885
US-20050090523-A1 2-(substituted phenyl)imidazo[1,2-a]pyridine compounds; use to treat disorders mediated by the histamine H3 receptor such as sleep disorders, attention deficit hyperactivity disorder, or Alzheimer's disease; 2-[4-[3-(Piperidino)propylamino]phenyl]-8-methylimidazo[1,2-a]pyridine for example HRH3, HRH4, HTR2C CYP2D6 681/4885MEN1 3966/4885KMT2A 57/4885
US-11639352-B2 Benzothiazole compounds for the treatment of autoimmune diseases SSB, BET1, HLA-DRB1 CYP2D6 1560/4885MEN1 328/4885KMT2A 963/4885
US-20020006934-A1 Phenyl-substituted imidazopyridines AADAC, DPP4, DPP3 CYP2D6 46/4885MEN1 4485/4885KMT2A 2545/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.