SCHEMBL28607435

SCHEMBL28607435

COc1ccc2c(c1)CC(=O)N2.Cc1cc(C)c(C(=O)O)[nH]1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 2/20 0.46
PDE3A Q14432 2/20 0.46
SRC P12931 1/20 0.44
GAA P10253 3/20 0.43
GRIA1 P42261 2/20 0.41
CACNG8 Q8WXS5 2/20 0.41
RET P07949 1/20 0.41
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41
ALPL P05186 1/20 0.41
CLK1 P49759 1/20 0.41
KMT2A Q03164 1/20 0.41
HSD17B10 Q99714 1/20 0.41
MAOB P27338 4/20 0.40
MAOA P21397 1/20 0.40
NPC1 O15118 1/20 0.39
ALDH1A1 P00352 1/20 0.39
AHR P35869 1/20 0.39
PKM P14618 1/20 0.38
CRBN Q96SW2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28597906 0.91 EIF2AK2 (0.50) PDE3BPDE3ASRCRETKDM4E
SCHEMBL29016221 0.83 AHR (0.47) PDE3BPDE3AGAAGRIA1CACNG8
SCHEMBL31040124 0.81 PDE3B (0.66) PDE3BPDE3ASRCGAAGRIA1
SCHEMBL20214 0.81 PDE3B (0.66) PDE3BPDE3ASRCGAAGRIA1
Trifluoroacetic Acid SCHEMBL29921460 0.78 PDE3B (0.52) PDE3BPDE3ASRCGAAMAOB
SCHEMBL3285782 0.76 NPC1 (0.59) PDE3BPDE3ASRCGAAGRIA1
SCHEMBL29016211 0.75 CRBN (0.53) GRIA1CACNG8AHRCRBNEIF2AK2
SCHEMBL6981292 0.71 AHR (0.51) PDE3BPDE3AGAAGRIA1CACNG8
SCHEMBL155069 0.71 PDE3B (0.62) PDE3BPDE3ASRCGAAGRIA1
SCHEMBL11469106 0.71 GAA (0.50) PDE3BPDE3AGAAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113181362-B Medicament for preventing and/or treating amyotrophic lateral sclerosis 国立大学法人京都大学 2023-06-13 CN disclosed
CN-113181362-A Agent for preventing and/or treating amyotrophic lateral sclerosis 国立大学法人京都大学 2021-07-30 CN disclosed