SCHEMBL286088

SCHEMBL286088

Cc1onc(-c2ccc(F)cc2)c1CNc1cc(C(=O)OC(C)C(N)=O)[nH]n1

nearest known ligand 0.54

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GABRA5 P31644 16/20 0.54
ENPP2 Q13822 1/20 0.42
KDM4E B2RXH2 1/20 0.40
THRB P10828 1/20 0.40
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL286172 0.87 GABRA5 (0.66) GABRA5ENPP2THRB
SCHEMBL286195 0.86 GABRA5 (0.56) GABRA5ENPP2KDM4ETHRB
SCHEMBL285983 0.84 GABRA5 (0.68) GABRA5ENPP2KDM4E
SCHEMBL286204 0.83 GABRA5 (0.57) GABRA5ENPP2KDM4ETHRB
SCHEMBL286153 0.83 GABRA5 (0.52) GABRA5ENPP2THRBKMT2A
SCHEMBL286087 0.80 GABRA5 (0.57) GABRA5ENPP2KDM4E
SCHEMBL286566 0.80 GABRA5 (0.53) GABRA5ENPP2KDM4ETHRB
SCHEMBL286432 0.80 GABRA5 (0.54) GABRA5ENPP2KDM4ETHRB
SCHEMBL286286 0.79 KDM4E (0.39) GABRA5KDM4EKMT2A
SCHEMBL286395 0.77 GABRA5 (0.58) GABRA5ENPP2KDM4ETHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427455-A1 ISOXAZOLE-PYRAZOLE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2012-03-14 EP disclosed