SCHEMBL286286

SCHEMBL286286

Cc1onc(-c2ccc(F)cc2)c1C=Cc1cc(C(=O)OC(C)C(N)=O)[nH]n1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.39
LMNA P02545 1/20 0.36
PTGS2 P35354 2/20 0.36
GABRA5 P31644 5/20 0.34
BACE1 P56817 2/20 0.34
KMT2A Q03164 2/20 0.34
POLB P06746 1/20 0.33
CASP6 P55212 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
ALPL P05186 1/20 0.33
FPR2 P25090 1/20 0.33
SCN9A Q15858 1/20 0.33
BTK Q06187 1/20 0.33
GPBAR1 Q8TDU6 1/20 0.33
MEN1 O00255 1/20 0.33
GAA P10253 1/20 0.33
RET P07949 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL285882 0.86 KDM4E (0.43) KDM4ELMNAPTGS2GABRA5BACE1
SCHEMBL285881 0.86 KDM4E (0.43) KDM4ELMNAPTGS2GABRA5BACE1
SCHEMBL286207 0.86 LMNA (0.46) KDM4ELMNAPTGS2GABRA5POLB
SCHEMBL286206 0.86 LMNA (0.46) KDM4ELMNAPTGS2GABRA5POLB
SCHEMBL286004 0.83 GABRA5 (0.46) KDM4ELMNAPTGS2GABRA5BACE1
SCHEMBL286002 0.83 GABRA5 (0.46) KDM4ELMNAPTGS2GABRA5BACE1
SCHEMBL286110 0.82 ALPL (0.48) KDM4ELMNAPTGS2GABRA5BACE1
SCHEMBL286109 0.82 ALPL (0.48) KDM4ELMNAPTGS2GABRA5BACE1
SCHEMBL286155 0.81 LMNA (0.36) LMNAPTGS2GABRA5BACE1KMT2A
SCHEMBL286088 0.79 GABRA5 (0.54) KDM4EGABRA5KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427455-A1 ISOXAZOLE-PYRAZOLE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2012-03-14 EP disclosed