SCHEMBL28608939

SCHEMBL28608939

COc1ccc(C2(Cn3cncn3)OCC(C)(C)CO2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.47
MAPT P10636 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
HSP90AA1 P07900 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
CYP19A1 P11511 4/20 0.38
CYP3A4 P08684 7/20 0.38
THRB P10828 1/20 0.38
CYP1A2 P05177 3/20 0.35
CYP2C9 P11712 3/20 0.35
CYP2C19 P33261 3/20 0.35
CYP2D6 P10635 2/20 0.35
TSHR P16473 1/20 0.34
GRIN1 Q05586 1/20 0.34
GRIN2B Q13224 1/20 0.34
CHRNA1 P02708 1/20 0.34
CHRNG P07510 1/20 0.34
CHRNB1 P11230 1/20 0.34
CHRNB2 P17787 1/20 0.34
CHRNB4 P30926 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11541496 0.89 ALDH1A1 (0.50) ALDH1A1MAPTSMN1; SMN2HSP90AA1NPSR1
SCHEMBL11542005 0.86 ALDH1A1 (0.48) ALDH1A1MAPTSMN1; SMN2HSP90AA1NPSR1
SCHEMBL9201064 0.81 ALDH1A1 (0.50) ALDH1A1MAPTSMN1; SMN2HSP90AA1NPSR1
SCHEMBL11547531 0.80 HSP90AA1 (0.56) ALDH1A1MAPTSMN1; SMN2HSP90AA1NPSR1
SCHEMBL9203493 0.78 ALDH1A1 (0.49) ALDH1A1MAPTSMN1; SMN2HSP90AA1NPSR1
SCHEMBL11543994 0.75 LMNA (0.42) ALDH1A1MAPTSMN1; SMN2HSP90AA1NPSR1
SCHEMBL10597473 0.75 ALDH1A1 (0.46) ALDH1A1MAPTSMN1; SMN2HSP90AA1NPSR1
SCHEMBL9457977 0.74 KDM4E (0.46) ALDH1A1MAPTSMN1; SMN2HSP90AA1NPSR1
SCHEMBL11547515 0.74 HSP90AA1 (0.63) ALDH1A1MAPTSMN1; SMN2HSP90AA1NPSR1
SCHEMBL9087052 0.74 ALDH1A1 (0.45) ALDH1A1MAPTSMN1; SMN2HSP90AA1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113234066-A Propiconazole-like compound and preparation method and application thereof 浙江工业大学 2021-08-10 CN disclosed