SCHEMBL28610469

SCHEMBL28610469

COC(=O)C(COC1CCN(C(=O)OCc2ccccc2)CC1)NC(=O)OC(C)(C)C

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.52
YAP1 P46937 2/20 0.51
SMN1; SMN2 Q16637 3/20 0.50
NPC1 O15118 2/20 0.50
RAB9A P51151 2/20 0.50
KLK7 P49862 2/20 0.49
KLK5 Q9Y337 2/20 0.49
MAPK1 P28482 1/20 0.48
PPARA Q07869 1/20 0.47
CYP2C19 P33261 1/20 0.47
KMT2A Q03164 2/20 0.47
CTSL P07711 1/20 0.47
ITGB3 P05106 1/20 0.46
ITGA2B P08514 1/20 0.46
CTSS P25774 1/20 0.45
SYK P43405 1/20 0.45
GAA P10253 1/20 0.45
PDE4B Q07343 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28610465 0.93 PPARA (0.55) HTTYAP1SMN1; SMN2NPC1RAB9A
SCHEMBL28610466 0.93 PPARA (0.55) HTTYAP1SMN1; SMN2NPC1RAB9A
SCHEMBL22433813 0.93 YAP1 (0.56) HTTYAP1SMN1; SMN2NPC1RAB9A
SCHEMBL31646670 0.90 KLK7 (0.50) HTTYAP1KLK7KLK5MAPK1
SCHEMBL27406331 0.89 ITGB3 (0.51) HTTYAP1KLK7KLK5MAPK1
SCHEMBL29968272 0.87 YAP1 (0.57) HTTYAP1SMN1; SMN2NPC1RAB9A
SCHEMBL12025774 0.87 YAP1 (0.57) HTTYAP1SMN1; SMN2NPC1RAB9A
SCHEMBL29189817 0.87 YAP1 (0.57) HTTYAP1SMN1; SMN2NPC1RAB9A
SCHEMBL12025747 0.87 YAP1 (0.57) HTTYAP1SMN1; SMN2NPC1RAB9A
SCHEMBL24979440 0.86 YAP1 (0.54) HTTYAP1MAPK1PPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107098871-B Phenyl propionamide derivative, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2021-07-02 CN disclosed