SCHEMBL28612669

SCHEMBL28612669

C[C@]12CON(Cc3ccccc3)[C@H]1CN(C(=O)O)C2

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AMPD2 Q01433 2/20 0.37
GAA P10253 1/20 0.37
CYP2D6 P10635 4/20 0.35
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
ALDH1A1 P00352 3/20 0.35
LMNA P02545 1/20 0.35
TMEM97 Q5BJF2 1/20 0.35
SIGMAR1 Q99720 1/20 0.35
TSHR P16473 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
S1PR1 P21453 1/20 0.35
S1PR5 Q9H228 1/20 0.35
BRD4 O60885 2/20 0.34
SIRT1 Q96EB6 1/20 0.34
GRM6 O15303 1/20 0.34
CYP3A4 P08684 1/20 0.34
HSD11B1 P28845 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21682573 1.00 AMPD2 (0.37) AMPD2GAACYP2D6MEN1KMT2A
SCHEMBL21682344 0.87 L3MBTL1 (0.41) GAAMEN1KMT2AALDH1A1SIGMAR1
SCHEMBL29422875 0.87 L3MBTL1 (0.41) GAAMEN1KMT2AALDH1A1SIGMAR1
SCHEMBL20397168 0.73 GAA (0.46) GAACYP2D6MEN1KMT2AALDH1A1
SCHEMBL6324844 0.69 GAA (0.51) GAACYP2D6MEN1KMT2AALDH1A1
SCHEMBL20399590 0.68 DRD4 (0.44) GAACYP2D6MEN1KMT2AALDH1A1
SCHEMBL20399589 0.68 DRD4 (0.44) GAACYP2D6MEN1KMT2AALDH1A1
SCHEMBL21819742 0.66 RECQL (0.43) MEN1KMT2AALDH1A1LMNATSHR
SCHEMBL28623607 0.66 RECQL (0.43) MEN1KMT2AALDH1A1LMNATSHR
SCHEMBL5029764 0.66 AMPD2 (0.36) AMPD2GAACYP2D6MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113272309-B Tricyclic inhibitors of hepatitis b virus 圣拉斐尔医院有限公司 2024-02-23 CN disclosed
CN-114555608-A Oxamide substituted tricyclic inhibitors of hepatitis b virus 分子遗传国家研究所(INGM) 2022-05-27 CN disclosed
CN-113272309-A Tricyclic inhibitors of hepatitis B virus 圣拉斐尔医院有限公司 2021-08-17 CN disclosed