SCHEMBL28612840

SCHEMBL28612840

O=C(O)N1CCN(Cc2ccc(OC(F)F)cc2)CC1COC(F)F

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.39
CCR1 P32246 1/20 0.39
S1PR5 Q9H228 4/20 0.39
SIGMAR1 Q99720 1/20 0.39
S1PR1 P21453 1/20 0.39
DPP4 P27487 1/20 0.39
DPP7 Q9UHL4 1/20 0.39
CHRM4 P08173 1/20 0.39
KMT2A Q03164 1/20 0.39
CA1 P00915 2/20 0.38
CA2 P00918 2/20 0.38
CA4 P22748 2/20 0.38
CA9 Q16790 2/20 0.38
ALDH1A1 P00352 2/20 0.38
HTT P42858 1/20 0.38
AGTR2 P50052 1/20 0.38
FAAH O00519 1/20 0.38
KCNH2 Q12809 1/20 0.37
MCHR1 Q99705 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28612839 1.00 POLB (0.39) POLBCCR1S1PR5SIGMAR1S1PR1
SCHEMBL28624276 0.86 LMNA (0.49) SIGMAR1KMT2AALDH1A1FAAH
SCHEMBL31599262 0.86 POLB (0.38) POLBCCR1S1PR5SIGMAR1S1PR1
SCHEMBL28577987 0.81 LTA4H (0.40) POLBCHRM4KMT2AALDH1A1HTT
SCHEMBL28577985 0.81 LTA4H (0.40) POLBCHRM4KMT2AALDH1A1HTT
SCHEMBL28610910 0.77 GPR6 (0.35) POLBS1PR5SIGMAR1S1PR1CHRM4
SCHEMBL28610908 0.77 GPR6 (0.35) POLBS1PR5SIGMAR1S1PR1CHRM4
SCHEMBL28622444 0.75 KCNH2 (0.40) KMT2AAGTR2FAAHKCNH2
SCHEMBL28612855 0.74 SLC6A4 (0.31)
SCHEMBL28612857 0.74 SLC6A4 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113072546-A Five-membered heteroaromatic derivative and preparation method and application thereof 广东东阳光药业有限公司 2021-07-06 CN disclosed