SCHEMBL28577985

SCHEMBL28577985

O=C(O)c1ccc(N2CCN(Cc3ccc(OC(F)F)cc3)C[C@H]2COC(F)F)cc1

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 6/20 0.40
CHRM4 P08173 1/20 0.40
ALDH1A1 P00352 3/20 0.39
HTT P42858 1/20 0.39
CPT1A P50416 1/20 0.38
CPT1B Q92523 1/20 0.38
KMT2A Q03164 3/20 0.38
MEN1 O00255 2/20 0.37
POLB P06746 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
MRGPRX4 Q96LA9 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28577987 1.00 LTA4H (0.40) LTA4HCHRM4ALDH1A1HTTCPT1A
SCHEMBL23632390 0.87 LMNA (0.45) LTA4HALDH1A1POLBL3MBTL1
SCHEMBL23632389 0.87 LMNA (0.45) LTA4HALDH1A1POLBL3MBTL1
SCHEMBL28612839 0.81 POLB (0.39) CHRM4ALDH1A1HTTKMT2APOLB
SCHEMBL28612840 0.81 POLB (0.39) CHRM4ALDH1A1HTTKMT2APOLB
SCHEMBL28610910 0.80 GPR6 (0.35) CHRM4KMT2APOLB
SCHEMBL28610908 0.80 GPR6 (0.35) CHRM4KMT2APOLB
SCHEMBL28593230 0.78 RORC (0.43)
SCHEMBL28593228 0.78 RORC (0.43)
SCHEMBL30075126 0.77 MEN1 (0.49) ALDH1A1KMT2AMEN1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113072521-B ROR gamma t inhibitor and application thereof in medicines 广东东阳光药业股份有限公司 2024-04-05 CN disclosed
CN-113072521-A ROR gamma t inhibitor and application thereof in medicine 广东东阳光药业有限公司 2021-07-06 CN disclosed