SCHEMBL28612909

SCHEMBL28612909

CN(C)C(=O)C1Cc2ccccc2O1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.54
TSHR P16473 1/20 0.54
CYP2D6 P10635 4/20 0.49
OPRK1 P41145 4/20 0.49
NFKB1 P19838 1/20 0.47
NFKB2 Q00653 1/20 0.47
RELA Q04206 1/20 0.47
AOC2 O75106 5/20 0.47
MAOA P21397 5/20 0.47
MAOB P27338 5/20 0.47
DAO P14920 1/20 0.47
HDAC6 Q9UBN7 2/20 0.44
HDAC3 O15379 1/20 0.44
HDAC4 P56524 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC7 Q8WUI4 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC10 Q969S8 1/20 0.44
HDAC11 Q96DB2 1/20 0.44
HDAC8 Q9BY41 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2153055 0.84 HPGD (0.49) HPGDTSHRCYP2D6OPRK1NFKB1
SCHEMBL2152568 0.81 HPGD (0.58) HPGDTSHRCYP2D6OPRK1NFKB1
SCHEMBL27730852 0.80 HPGD (0.61) HPGDTSHRNFKB1NFKB2RELA
SCHEMBL5847146 0.79 HPGD (0.64) HPGDTSHRCYP2D6OPRK1NFKB1
SCHEMBL29974170 0.79 HPGD (0.59) HPGDTSHRNFKB1NFKB2RELA
SCHEMBL860446 0.79 HPGD (0.59) HPGDTSHRNFKB1NFKB2RELA
SCHEMBL5109501 0.79 HPGD (0.64) HPGDTSHRCYP2D6OPRK1NFKB1
SCHEMBL1519327 0.79 HPGD (0.64) HPGDTSHRCYP2D6OPRK1NFKB1
SCHEMBL2103264 0.78 POLB (0.42) HPGDTSHRCYP2D6OPRK1NFKB1
SCHEMBL15796618 0.78 GLS (0.47) CYP2D6OPRK1GLS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107660205-B Heterocyclic compounds as LSD1 inhibitors 因赛特公司 2021-08-27 CN claimed
CN-107660205-B Heterocyclic compounds as LSD1 inhibitors 因赛特公司 2021-08-27 CN disclosed