SCHEMBL28614756

SCHEMBL28614756

CN(C)c1ccc(C(=O)NC(CCC(=O)O)C(=O)O)s1

nearest known ligand 0.55

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TYMS P04818 6/20 0.55
FOLR1 P15328 2/20 0.55
DHFR P00374 1/20 0.55
FOLR2 P14207 1/20 0.55
SLC19A1 P41440 1/20 0.55
EHMT2 Q96KQ7 1/20 0.55
SLC46A1 Q96NT5 1/20 0.55
LMNA P02545 1/20 0.55
CA2 P00918 2/20 0.48
CA1 P00915 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28614753 1.00 TYMS (0.55) TYMSFOLR1DHFRFOLR2SLC19A1
SCHEMBL27559568 0.82 CA2 (0.53) FOLR1FOLR2SLC19A1SLC46A1CA2
SCHEMBL9600674 0.81 CA2 (0.52) TYMSFOLR1FOLR2SLC19A1SLC46A1
SCHEMBL9600688 0.81 CA2 (0.52) TYMSFOLR1FOLR2SLC19A1SLC46A1
SCHEMBL27513231 0.80 TYMS (0.55) TYMSFOLR1DHFRFOLR2SLC19A1
SCHEMBL9829787 0.80 TYMS (0.55) TYMSFOLR1DHFRFOLR2SLC19A1
SCHEMBL9829799 0.80 TYMS (0.55) TYMSFOLR1DHFRFOLR2SLC19A1
SCHEMBL9379643 0.78 TYMS (0.56) TYMSFOLR1DHFRFOLR2SLC19A1
SCHEMBL9514889 0.78 TYMS (0.55) TYMS
SCHEMBL9379640 0.78 TYMS (0.56) TYMSFOLR1DHFRFOLR2SLC19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117327060-A Preparation method of intermediate impurity of raltitrexed 无锡紫杉药业股份有限公司 2024-01-02 CN disclosed
CN-109280044-B Raltitrexed impurity C and preparation and application thereof 南京正大天晴制药有限公司 2021-04-02 CN disclosed