SCHEMBL28614947

SCHEMBL28614947

O=C(CCCCCCNC(=O)C1CCc2[nH]c3ccccc3c2C1)NO

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 12/20 0.52
HDAC6 Q9UBN7 10/20 0.52
HDAC2 Q92769 10/20 0.47
HDAC3 O15379 8/20 0.47
HDAC4 P56524 8/20 0.47
HDAC7 Q8WUI4 8/20 0.47
HDAC10 Q969S8 8/20 0.47
HDAC11 Q96DB2 8/20 0.47
HDAC8 Q9BY41 8/20 0.47
HDAC9 Q9UKV0 8/20 0.47
HDAC5 Q9UQL6 8/20 0.47
ACHE P22303 1/20 0.44
NR2E1 Q9Y466 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28617694 0.91 HDAC1 (0.53) HDAC1HDAC6HDAC2HDAC3HDAC4
SCHEMBL28603643 0.87 KDM4E (0.44) ACHENR2E1
SCHEMBL14476893 0.83 ACHE (0.59) HDAC1HDAC6HDAC2HDAC3HDAC4
SCHEMBL4725539 0.82 KMT2A (0.49) NR2E1
SCHEMBL28618175 0.78 KDM4E (0.47) ACHE
SCHEMBL28617480 0.76 KMT2A (0.73) HDAC1HDAC6HDAC2HDAC3HDAC4
SCHEMBL14476888 0.75 ACHE (0.65) HDAC1HDAC6HDAC8ACHE
SCHEMBL28614964 0.74 HDAC6 (0.78) HDAC1HDAC6
SCHEMBL24479988 0.73 NPSR1 (0.47) NR2E1
SCHEMBL5956886 0.73 HDAC1 (0.66) HDAC1HDAC6HDAC2HDAC3HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113121527-A Tricyclic compound and use thereof 上海辉启生物医药科技有限公司 2021-07-16 CN disclosed