SCHEMBL4725539

SCHEMBL4725539

CCCNC(=O)C1CCc2[nH]c3ccccc3c2C1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.49
NR2E1 Q9Y466 1/20 0.49
SLC2A1 P11166 1/20 0.46
HSD17B10 Q99714 3/20 0.46
KDM4E B2RXH2 2/20 0.46
CYP1A2 P05177 2/20 0.46
CYP2D6 P10635 2/20 0.46
CYP2C9 P11712 2/20 0.46
CYP2C19 P33261 2/20 0.46
HPGD P15428 2/20 0.46
ALDH1A1 P00352 1/20 0.46
GAA P10253 1/20 0.46
MAPT P10636 1/20 0.46
ALOX15 P16050 1/20 0.46
MAPK1 P28482 1/20 0.45
TRPM8 Q7Z2W7 1/20 0.44
MTNR1A P48039 1/20 0.44
MTNR1B P49286 1/20 0.44
TP53 P04637 1/20 0.44
CYP19A1 P11511 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28603643 0.83 KDM4E (0.44) KMT2ANR2E1HSD17B10KDM4ECYP1A2
SCHEMBL28614947 0.82 HDAC1 (0.52) NR2E1
SCHEMBL4763963 0.80 NR2E1 (0.52) KMT2ANR2E1SLC2A1HSD17B10KDM4E
SCHEMBL24479988 0.79 NPSR1 (0.47) NR2E1HSD17B10KDM4EALDH1A1MAPK1
SCHEMBL30523189 0.79 KDM4E (0.63) KMT2ANR2E1HSD17B10KDM4ECYP1A2
SCHEMBL30523188 0.79 KDM4E (0.63) KMT2ANR2E1HSD17B10KDM4ECYP1A2
SCHEMBL4728062 0.79 KDM4E (0.63) KMT2ANR2E1HSD17B10KDM4ECYP1A2
SCHEMBL31078247 0.79 KDM4E (0.64) KMT2ANR2E1SLC2A1HSD17B10KDM4E
SCHEMBL4727252 0.79 KDM4E (0.64) KMT2ANR2E1SLC2A1HSD17B10KDM4E
SCHEMBL4903024 0.79 NR2E1 (0.64) NR2E1HSD17B10KDM4ECYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008021745-A2 HEPATITIS C VIRUS ENTRY INHIBITORS ITHERX PHARMACEUTICALS, INC. (US) 2008-02-21 WO disclosed