SCHEMBL28615500

SCHEMBL28615500

O=C(O)c1ccc(CI)cc1CI

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 1/20 0.41
CTSB P07858 1/20 0.41
MMP9 P14780 1/20 0.41
DNMT1 P26358 1/20 0.41
DNMT3B Q9UBC3 1/20 0.41
DNMT3L Q9UJW3 1/20 0.41
DNMT3A Q9Y6K1 1/20 0.41
TSHR P16473 3/20 0.41
ALDH1A1 P00352 2/20 0.40
CDC25B P30305 1/20 0.40
CASP6 P55212 1/20 0.40
RCE1 Q9Y256 1/20 0.40
DCLRE1A Q6PJP8 1/20 0.40
DCLRE1B Q9H816 1/20 0.40
CYP1A2 P05177 1/20 0.39
PTPN1 P18031 2/20 0.39
PTPN2 P17706 1/20 0.39
PTPN6 P29350 1/20 0.39
LCK P06239 2/20 0.38
HNF4A P41235 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27704208 0.80 TSHR (0.33) KLKB1CTSBMMP9DNMT1DNMT3B
SCHEMBL5713415 0.80 PPARA (0.36) KLKB1CTSBMMP9DNMT1DNMT3B
SCHEMBL2226926 0.80 PPARA (0.56) KLKB1CTSBMMP9DNMT1DNMT3B
SCHEMBL17049075 0.80 EPHX2 (0.47) KLKB1CTSBMMP9DNMT1DNMT3B
SCHEMBL27716557 0.78 ALDH1A1 (0.52) KLKB1CTSBMMP9DNMT1DNMT3B
SCHEMBL7025446 0.78 NR1H4 (0.50) KLKB1CTSBMMP9DNMT1DNMT3B
SCHEMBL27496275 0.78 TSHR (0.57) KLKB1CTSBMMP9DNMT1DNMT3B
SCHEMBL13806629 0.78 KEAP1 (0.48) TSHRALDH1A1DCLRE1ADCLRE1BCYP1A2
SCHEMBL27336883 0.76 KLKB1 (0.71) KLKB1CTSBMMP9DNMT1DNMT3B
SCHEMBL8479634 0.74 CA12 (0.45) KLKB1CTSBMMP9DNMT1DNMT3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113226377-A Antibody drug conjugates comprising an eltrinastine derivative 法马马有限公司 2021-08-06 CN disclosed