SCHEMBL28616385

SCHEMBL28616385

N#Cc1cc(F)c(OC(F)F)cc1OC(N)=O

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 4/20 0.37
CYP2D6 P10635 3/20 0.37
SLC6A2 P23975 3/20 0.37
SLC6A4 P31645 3/20 0.37
CYP11B2 P19099 1/20 0.33
KMT2A Q03164 1/20 0.31
SLC22A12 Q96S37 1/20 0.30
S1PR1 P21453 1/20 0.30
S1PR3 Q99500 1/20 0.30
TRPV4 Q9HBA0 1/20 0.30
F11 P03951 1/20 0.30
KLKB1 P03952 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29177252 0.83 KMT2A (0.36) KMT2AS1PR3
SCHEMBL28586926 0.83 CYP2D6 (0.33) NOS2CYP2D6SLC6A2SLC6A4F11
SCHEMBL28603822 0.78 VCAM1 (0.37) KMT2AF11KLKB1
SCHEMBL21996464 0.75 KHK (0.38) NOS2CYP2D6SLC6A2SLC6A4TRPV4
SCHEMBL29177363 0.75 BACE1 (0.33) KMT2A
SCHEMBL3532342 0.74 CYP2D6 (0.40) NOS2CYP2D6SLC6A2SLC6A4CYP11B2
SCHEMBL28246635 0.74 FFAR1 (0.49) CYP11B2KMT2ASLC22A12
SCHEMBL21996274 0.73 KMT2A (0.39) NOS2CYP2D6SLC6A2SLC6A4KMT2A
SCHEMBL24196446 0.72 NOS2 (0.40) NOS2CYP2D6SLC6A2SLC6A4CYP11B2
SCHEMBL28738823 0.72 ALDH1A1 (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113329791-A 9-substituted amino-triazoloquinazoline derivatives as adenosine receptor antagonists, pharmaceutical compositions and uses thereof 默沙东公司 2021-08-31 CN disclosed