SCHEMBL28616833

SCHEMBL28616833

CCc1csc2c(S(C)(=O)=O)ncnc12

nearest known ligand 0.32

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 4/20 0.32
PDE4B Q07343 1/20 0.30
PDE7A Q13946 1/20 0.30
MAPK1 P28482 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30808298 1.00 GPR119 (0.32) GPR119PDE4BPDE7AMAPK1
SCHEMBL28613438 0.85
SCHEMBL15751094 0.80 GPR35 (0.31)
SCHEMBL30808281 0.77 PIP4K2C (0.42) GPR119PDE4BPDE7A
SCHEMBL28606328 0.77 PIP4K2C (0.42) GPR119PDE4BPDE7A
SCHEMBL19073526 0.75 CDC7 (0.41)
SCHEMBL28613381 0.73 PDPK1 (0.49) GPR119
SCHEMBL21823142 0.72 ALDH1A1 (0.36) PDE4BPDE7AMAPK1
SCHEMBL12505973 0.72 GPR119 (0.51) GPR119
SCHEMBL21823036 0.70 MAPK1 (0.47) GPR119MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113039182-B Inhibitors of YAP/TAZ-TEAD interactions and their use in cancer treatment 伊文蒂瓦公司 2024-02-20 CN disclosed
CN-113039182-A Inhibitors of YAP/TAZ-TEAD interaction and their use in cancer treatment 伊文蒂瓦公司 2021-06-25 CN disclosed