SCHEMBL28619610

SCHEMBL28619610

Cn1nc(C(C)(C)C)c2cc(Br)cnc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 1/20 0.40
GSK3B P49841 2/20 0.38
POLB P06746 1/20 0.32
SPR P35270 1/20 0.32
MAOB P27338 1/20 0.32
PDE1B Q01064 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
CHEK1 O14757 1/20 0.30
AURKA O14965 1/20 0.30
DAPK3 O43293 1/20 0.30
JAK2 O60674 1/20 0.30
MAP4K4 O95819 1/20 0.30
PAK4 O96013 1/20 0.30
ABL1 P00519 1/20 0.30
CSF1R P07333 1/20 0.30
RET P07949 1/20 0.30
IGF1R P08069 1/20 0.30
FGFR1 P11362 1/20 0.30
PDGFRA P16234 1/20 0.30
PRKACA P17612 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27259567 0.85 GSK3B (0.40) HSD17B10GSK3BPOLBMAOB
SCHEMBL29324752 0.81 GSK3B (0.39) GSK3BPOLBSPRHCRTR1HCRTR2
SCHEMBL18538040 0.80 HPGD (0.40) HSD17B10GSK3BPOLBSPRNPSR1
SCHEMBL25527223 0.80 GSK3B (0.38) GSK3BPOLBSPRHCRTR1HCRTR2
SCHEMBL18538049 0.78 ALDH1A1 (0.42) GSK3BPOLBMAOBNPSR1
SCHEMBL6952100 0.77 SPR (0.46) HSD17B10GSK3BPOLBSPRCHEK1
SCHEMBL30924204 0.77 SPR (0.46) HSD17B10GSK3BPOLBSPRCHEK1
SCHEMBL12703712 0.76 HSD17B10 (0.46) HSD17B10GSK3BPOLBSPRMAOB
SCHEMBL31149372 0.76 HSD17B10 (0.42) HSD17B10GSK3BPOLBSPRMAOB
SCHEMBL12703617 0.76 HSD17B10 (0.42) HSD17B10GSK3BPOLBSPRMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108602799-B Kinase inhibitor 上海复尚慧创医药研究有限公司 2021-08-03 CN disclosed